SCHEMBL13809253

SCHEMBL13809253

COc1ccc(OC)c2c1CCN(C(=O)c1ccccc1C(C)=O)C2c1cccc(Cl)c1Cl

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2C Q14957 1/20 0.43
POLB P06746 2/20 0.40
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
P2RX7 Q99572 5/20 0.37
ALDH1A1 P00352 1/20 0.37
HSD11B1 P28845 1/20 0.37
HHAT Q5VTY9 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809228 0.88 GRIN2C (0.43) GRIN2CABCB1ABCG2P2RX7HSD11B1
SCHEMBL13809007 0.86 GRIN2C (0.43) GRIN2CPOLBABCB1ABCG2P2RX7
SCHEMBL13809241 0.85 GRIN2C (0.41) GRIN2CABCB1ABCG2P2RX7ALDH1A1
SCHEMBL13809231 0.82 GRIN2C (0.39) GRIN2CABCB1ABCG2P2RX7
SCHEMBL13809234 0.80 GRIN2C (0.40) GRIN2CABCB1ABCG2MEN1KMT2A
SCHEMBL13809244 0.80 GRIN2C (0.36) GRIN2CPOLBALDH1A1HHATMEN1
SCHEMBL13809226 0.74 ABCG2 (0.39) GRIN2CABCB1ABCG2P2RX7HSD11B1
SCHEMBL13809251 0.71 GRIN2C (0.49) GRIN2CALDH1A1MEN1KMT2A
SCHEMBL13808738 0.67 MAPT (0.42)
SCHEMBL13809240 0.65 GRIN2C (0.54) GRIN2CMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed