SCHEMBL13809241

SCHEMBL13809241

COc1ccc(OC)c2c1CCN(C(=O)c1ccc(C)cc1C(=O)O)C2c1cccc(Cl)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2C Q14957 1/20 0.41
CMA1 P23946 1/20 0.38
P2RX7 Q99572 6/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ABCB1 P08183 2/20 0.36
ABCG2 Q9UNQ0 2/20 0.36
LMNA P02545 2/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
NPC1 O15118 1/20 0.35
MITF O75030 1/20 0.35
ALDH1A1 P00352 1/20 0.35
XBP1 P17861 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
F11 P03951 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809007 0.91 GRIN2C (0.43) GRIN2CCMA1P2RX7MEN1KMT2A
SCHEMBL13809253 0.85 GRIN2C (0.43) GRIN2CP2RX7MEN1KMT2AABCB1
SCHEMBL13809228 0.81 GRIN2C (0.43) GRIN2CP2RX7MEN1KMT2AABCB1
SCHEMBL13809244 0.79 GRIN2C (0.36) GRIN2CCMA1MEN1KMT2ALMNA
SCHEMBL13809234 0.78 GRIN2C (0.40) GRIN2CMEN1KMT2AABCB1ABCG2
SCHEMBL13809231 0.76 GRIN2C (0.39) GRIN2CP2RX7ABCB1ABCG2
SCHEMBL13809251 0.76 GRIN2C (0.49) GRIN2CMEN1KMT2ALMNANPC1
SCHEMBL13809243 0.75 KIF11 (0.53) GRIN2CP2RX7MEN1KMT2ALMNA
SCHEMBL10025894 0.71 MAPT (0.41) MEN1KMT2ALMNATP53MAPT
SCHEMBL13809019 0.66 GRIN2C (0.44) GRIN2CMEN1KMT2ALMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed