SCHEMBL13809376

SCHEMBL13809376

CC(C)(C)OC(=O)N1CCC(NC(=O)c2ccc3[nH]c4c(c3c2)CN(C(=O)CCc2ccccc2)CC4)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.45
MAPT P10636 6/20 0.43
MAPK1 P28482 5/20 0.43
POLB P06746 3/20 0.43
NPSR1 Q6W5P4 3/20 0.43
GAA P10253 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
GPR55 Q9Y2T6 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 5/20 0.42
CASP1 P29466 2/20 0.42
ATM Q13315 2/20 0.42
KDM4E B2RXH2 2/20 0.42
HSD17B10 Q99714 1/20 0.42
NTSR1 P30989 1/20 0.41
CASP7 P55210 1/20 0.41
USP30 Q70CQ3 2/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL61054 0.89 L3MBTL1 (0.49) MAPTMAPK1POLBNPSR1GAA
SCHEMBL12264857 0.86 ROCK2 (0.52) TRPV1MAPK1GAAKMT2ATAAR1
SCHEMBL13809575 0.81 HDAC1 (0.59) MAPK1POLBNPSR1GAAMEN1
SCHEMBL61542 0.80 HDAC1 (0.52) POLBGAALMNAPARP1
SCHEMBL61089 0.79 HDAC1 (0.53) POLBGAAMEN1KMT2A
SCHEMBL62007 0.79 BRD3 (0.46) MAPTPOLBGAAKMT2AL3MBTL1
SCHEMBL16939031 0.79 POLB (0.43) MAPTMAPK1POLBNPSR1GAA
SCHEMBL62772 0.79 HDAC4 (0.45) POLBGAAMEN1KMT2AALDH1A1
SCHEMBL3312381 0.77 LMNA (0.57) MAPTMAPK1POLBGAAKMT2A
SCHEMBL62381 0.76 ROCK2 (0.51) MAPK1KMT2AATMLMNAPABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009076631-A1 CARBOXAMIDE, SULFONAMIDE AND AMINE COMPOUNDS FOR METABOLIC DISORDERS RIGEL PHARMACEUTICALS, INC. (US) 2009-06-18 WO disclosed