SCHEMBL13825501

SCHEMBL13825501

Bc1cccc(/C(=C/C)c2ccc(OC)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 6/20 0.46
PDE4B Q07343 6/20 0.46
PDE4C Q08493 6/20 0.46
PDE4D Q08499 6/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
CES2 O00748 3/20 0.42
CES1 P23141 3/20 0.42
KCNK9 Q9NPC2 1/20 0.40
MAOB P27338 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
NQO2 P16083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13825497 1.00 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL2284188 0.81 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL7862071 0.81 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL2284191 0.81 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6937356 0.80 ALDH1A1 (0.65) PDE4APDE4BPDE4CPDE4DKDM4E
Ammonia Solution, Strong SCHEMBL5700298 0.78 ALDH1A1 (0.63) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL14376098 0.77 CES2 (0.62) PDE4APDE4BPDE4CPDE4DCES2
SCHEMBL8270539 0.75 PDE4A (0.78) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL8270543 0.71 PDE4A (0.77) PDE4APDE4BPDE4CPDE4DNQO2
SCHEMBL8247682 0.71 SMN1; SMN2 (0.63) KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-B1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-11-14 EP disclosed