SCHEMBL13843809

SCHEMBL13843809

C#Cc1cnc(-c2ccccc2)n1CC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.54
HSD17B10 Q99714 1/20 0.54
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
NLRP3 Q96P20 1/20 0.40
TSHR P16473 1/20 0.39
ALDH1A1 P00352 3/20 0.37
MAPK14 Q16539 2/20 0.37
MAPT P10636 2/20 0.37
CHEK1 O14757 1/20 0.37
LIMK1 P53667 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HPGDS O60760 2/20 0.36
RAB9A P51151 2/20 0.35
GAA P10253 1/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13843808 0.78 HPGDS (0.50) KDM4EHSD17B10TLR7ALDH1A1MAPK14
SCHEMBL16193332 0.76 KDM4E (0.59) KDM4EHSD17B10ADORA3ADORA2AADORA2B
SCHEMBL28995656 0.75 LMNA (0.31) TSHRALDH1A1
SCHEMBL7913638 0.75 KDM4E (0.58) KDM4EHSD17B10ADORA3ADORA2AADORA2B
SCHEMBL4030659 0.71 KDM4E (0.54) KDM4EHSD17B10ADORA3ADORA2AADORA2B
SCHEMBL11768659 0.68 KDM4E (0.50) KDM4EHSD17B10ADORA2AADORA2BALDH1A1
SCHEMBL761987 0.67 KDM4E (0.49) KDM4EHSD17B10ADORA3ADORA2AADORA2B
SCHEMBL18419644 0.66 KDM4E (0.47) KDM4EHSD17B10TLR7TSHRALDH1A1
SCHEMBL19419968 0.66 KDM4E (0.47) KDM4EHSD17B10ADORA3ADORA2AADORA2B
SCHEMBL650528 0.66 TSHR (0.65) KDM4EHSD17B10ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531560-B2 Anti-cytokine heterocyclic compounds BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2009-05-12 US disclosed
US-7531560-B2 Anti-cytokine heterocyclic compounds BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2009-05-12 US disclosed