SCHEMBL13845000

SCHEMBL13845000

Nc1ccc(S(=O)(=O)N2CCC(Oc3ccccn3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MAPT P10636 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NAAA Q02083 1/20 0.47
USP5 P45974 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 1/20 0.45
HTR2C P28335 1/20 0.44
GRM4 Q14833 1/20 0.44
TP53 P04637 1/20 0.44
HTR2B P41595 1/20 0.44
PKM P14618 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
EPHX2 P34913 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
RORC P51449 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14095896 0.86 CYP19A1 (0.44) MEN1KMT2ASMN1; SMN2NPC1RAB9A
SCHEMBL3295631 0.80 NAAA (0.38) MEN1KMT2AMAPTSMN1; SMN2NAAA
SCHEMBL14095894 0.80 MAPT (0.63) MEN1KMT2AMAPTSMN1; SMN2USP5
SCHEMBL14095854 0.77 KMT2A (0.67) MEN1KMT2ASMN1; SMN2NPC1RAB9A
SCHEMBL13392256 0.74 LMNA (0.47) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL13489653 0.73 SMN1; SMN2 (0.68) MEN1KMT2AMAPTSMN1; SMN2USP5
SCHEMBL5898968 0.73 MMP2 (0.63) NAAANPC1RAB9AEPHX2
SCHEMBL11511360 0.73 KDM4E (0.76) MEN1KMT2AMAPTSMN1; SMN2PKM
SCHEMBL854850 0.72 MAPT (0.50) MEN1KMT2AMAPTSMN1; SMN2TP53
SCHEMBL29605026 0.72 AVPR1A (0.49) NAAAEPHX2KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056693-A1 NOVEL DERIVATIVES OF N, N'- 2, 4-DIANILINOPYRIMIDINES, PREPARATION THEREOF AS MEDICAMENTS PHARMACEUTICAL COMPOSITIONS AND IN PARTICULAR AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2009-05-07 WO disclosed
WO-2008099073-A1 N, N' -2, 4-DIANILINOPYRIMIDINES PREPARATION AND USE THEREOF AS IKK INHIBITORS PREPARATION AND TEH PHARMACUETICAL COMPOSITIONS THEREOF SANOFI-AVENTIS (FR) 2008-08-21 WO disclosed