SCHEMBL13876145

SCHEMBL13876145

COC(=O)[C@H](Cc1ccc(Oc2ccc(CC3SC(=S)NC3=O)cc2Cl)cc1)NCl

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.43
ALDH1A1 P00352 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
FFAR1 O14842 6/20 0.38
PPARG P37231 4/20 0.38
PTPN1 P18031 2/20 0.38
ACACB O00763 4/20 0.36
MPC2 O95563 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2C9 P11712 1/20 0.35
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13875697 0.92 ALDH1A1 (0.51) CA2ALDH1A1NPSR1FFAR1PPARG
SCHEMBL13875978 0.91 CA2 (0.48) CA2ALDH1A1NPSR1FFAR1PPARG
SCHEMBL13876150 0.91 CA2 (0.43) CA2ALDH1A1NPSR1FFAR1PPARG
SCHEMBL13866960 0.90 CA2 (0.43) CA2ALDH1A1NPSR1FFAR1PPARG
Hydrochloric Acid SCHEMBL3868269 0.89 CA2 (0.43) CA2ALDH1A1NPSR1FFAR1PPARG
SCHEMBL13875706 0.86 CA2 (0.48) CA2ALDH1A1NPSR1FFAR1PPARG
SCHEMBL13875929 0.83 PTPN1 (0.55) CA2ALDH1A1NPSR1FFAR1PPARG
SCHEMBL13875580 0.83 PTPN1 (0.46) CA2ALDH1A1NPSR1FFAR1PPARG
SCHEMBL13875705 0.82 CA2 (0.48) CA2FFAR1PPARGMPC2CYP2C8
SCHEMBL13908674 0.81 ALDH1A1 (0.51) CA2ALDH1A1NPSR1FFAR1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848700-B1 SALTS OF (S)-2-AMINO-3-{4-[4-(2,4-DIOXO-THIAZOLIDIN-5-YLMETHYL)-PHENOXY]-PHENYL}-PROPIONIC ACID AND ITS METHYL ESTER AS INTERLEUKIN INHIBITORS FOR THE TREATMENT OF OBESITY OR DIABETES BEXEL PHARMACEUTICALS INC (US) 2015-12-30 EP disclosed
US-7521465-B2 Diphenyl ether derivatives BEXEL PHARMACEUTICALS, INC. (US) 2009-04-21 US disclosed