SCHEMBL1387663

SCHEMBL1387663

CCCCCCCCCCc1ccc(N(CC(=O)O)C(=O)CN2CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 8/20 0.63
S1PR3 Q99500 5/20 0.47
S1PR4 O95977 3/20 0.47
S1PR5 Q9H228 3/20 0.47
ALDH1A1 P00352 2/20 0.45
S1PR2 O95136 2/20 0.43
RARB P10826 4/20 0.41
MEN1 O00255 1/20 0.41
RARA P10276 1/20 0.41
MAPT P10636 1/20 0.41
MTOR P42345 1/20 0.41
KMT2A Q03164 1/20 0.41
CYSLTR2 Q9NS75 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41
GSK3B P49841 1/20 0.41
SPHK1 Q9NYA1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9079285 0.98 S1PR1 (0.61) S1PR1S1PR3S1PR4S1PR5ALDH1A1
SCHEMBL9097562 0.89 S1PR1 (0.50) S1PR1S1PR3S1PR4S1PR5ALDH1A1
SCHEMBL20187534 0.78 CACNA2D1 (0.49) ALDH1A1
SCHEMBL177063 0.78 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5ALDH1A1
SCHEMBL9079952 0.77 MLYCD (0.40) ALDH1A1MEN1MAPTKMT2A
SCHEMBL9080067 0.74 ALDH1A1 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL9169757 0.74 ALDH1A1 (0.60) S1PR1S1PR3ALDH1A1S1PR2RARB
SCHEMBL9972487 0.74 ALDH1A1 (0.60) S1PR1S1PR3ALDH1A1S1PR2RARB
SCHEMBL27145122 0.74 S1PR1 (0.62) S1PR1S1PR3S1PR4S1PR5ALDH1A1
SCHEMBL15505725 0.71 SIGMAR1 (0.57) S1PR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-H08511809-A 1996-12-10 JP claimed
US-5573752-A Aromatic amide compounds and metal chelates thereof BRACCO INTERNATIONAL B.V. 1996-11-12 US claimed
WO-1995027705-A1 AROMATIC AMIDE COMPOUNDS AND METAL CHELATES THEREOF BRACCO INTERNATIONAL B.V. (NL) 1995-10-19 WO claimed
US-5573752-A Aromatic amide compounds and metal chelates thereof BRACCO INTERNATIONAL B.V. 1996-11-12 US disclosed