SCHEMBL13879

SCHEMBL13879

Cc1ccccc1-c1ccc2nc3c(cc2c1)C[C@H](C(=O)NC1CCCC(C)(C)C1)N3

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.44
ABL1 P00519 2/20 0.39
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14273 0.81 BACE1 (0.41) BACE1ABL1
SCHEMBL14210 0.78 BACE1 (0.41) BACE1ABL1
SCHEMBL9177 0.75 BACE1 (0.76) BACE1
SCHEMBL14321887 0.75 BACE1 (0.76) BACE1
SCHEMBL9869 0.74 BACE1 (0.80) BACE1
SCHEMBL13984 0.71 GRM5 (0.39) BACE1
SCHEMBL13664 0.63 BACE1 (0.57) BACE1ABL1
SCHEMBL14324803 0.62 BACE1 (0.83) BACE1
SCHEMBL11567 0.62 BACE1 (0.83) BACE1
SCHEMBL21739921 0.61 EPHX1 (0.49) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063233-A1 AMINO HETEROARYL COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2011-05-26 WO disclosed