SCHEMBL13984

SCHEMBL13984

O=C(NC1CCOC2(CCC2)C1)C1Cc2cc3cc(-c4cccc(Cl)c4)ccc3nc2N1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.39
CNR2 P34972 4/20 0.36
NPR1 P16066 1/20 0.36
BACE1 P56817 2/20 0.34
SMO Q99835 1/20 0.34
NPC1 O15118 3/20 0.33
RAB9A P51151 2/20 0.33
MAP4K4 O95819 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9354 0.75 BACE1 (0.62) GRM5BACE1
SCHEMBL14273 0.65 BACE1 (0.41) BACE1
SCHEMBL8662 0.65 BACE1 (0.75) BACE1
SCHEMBL764562 0.56 RAB9A (0.47) NPC1RAB9A
SCHEMBL31071537 0.55 ALDH1A1 (0.30)
SCHEMBL10287832 0.55 ABL1 (0.73)
SCHEMBL21739908 0.55 SMYD3 (0.39) CNR2SMONPC1RAB9A
SCHEMBL14226166 0.54 CNR2 (1.00) CNR2NPC1RAB9A
SCHEMBL31332809 0.53 SLC6A4 (0.46) GRM5NPC1RAB9A
SCHEMBL27162363 0.53 PDE4A (0.57) CNR2BACE1RAB9APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063233-A1 AMINO HETEROARYL COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2011-05-26 WO disclosed