SCHEMBL13880941

SCHEMBL13880941

COc1cc(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)ccc1N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.58
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
POLB P06746 1/20 0.57
BTK Q06187 1/20 0.56
KIT P10721 2/20 0.55
PKM P14618 1/20 0.55
LMNA P02545 2/20 0.55
ALDH1A1 P00352 2/20 0.55
HSD17B10 Q99714 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
USP2 O75604 1/20 0.55
MAPT P10636 1/20 0.55
HPGD P15428 1/20 0.55
ABCB1 P08183 2/20 0.54
ABCG2 Q9UNQ0 2/20 0.54
INSR P06213 1/20 0.54
ALK Q9UM73 1/20 0.54
HIF1A Q16665 1/20 0.53
EPAS1 Q99814 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12345537 0.88 NPC1 (0.62) KMT2ANPC1RAB9APOLBBTK
SCHEMBL13880860 0.82 ALK (0.56) LMNAALDH1A1SMN1; SMN2MAPTABCB1
SCHEMBL28668646 0.82 PKM (0.79) KMT2ANPC1RAB9ABTKPKM
SCHEMBL15651745 0.82 BTK (0.65) KMT2ANPC1RAB9APOLBBTK
SCHEMBL15381993 0.82 ALDH1A1 (0.64) KMT2ANPC1RAB9ABTKKIT
SCHEMBL22017243 0.82 KMT2A (0.57) KMT2ANPC1RAB9APOLBBTK
SCHEMBL21400972 0.80 NPC1 (0.79) KMT2ANPC1RAB9ABTKKIT
SCHEMBL846560 0.79 BTK (0.65) NPC1RAB9ABTKKITALDH1A1
SCHEMBL31436860 0.79 BTK (0.65) NPC1RAB9ABTKKITALDH1A1
SCHEMBL12426361 0.79 KMT2A (0.65) KMT2APOLBSMN1; SMN2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2564850-A1 Polo-like kinase inhibitors Takeda Pharmaceutical Company Limited (JP) 2013-03-06 EP disclosed
WO-2009042711-A1 POLO-LIKE KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed