SCHEMBL22017243

SCHEMBL22017243

CCC(=O)Nc1cc(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)ccc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.57
EGFR P00533 2/20 0.55
LMNA P02545 5/20 0.54
ALDH1A1 P00352 3/20 0.54
HPGD P15428 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
USP2 O75604 1/20 0.54
MAPT P10636 1/20 0.54
HSD17B10 Q99714 1/20 0.54
WNT3A P56704 1/20 0.54
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
POLB P06746 1/20 0.53
BTK Q06187 1/20 0.53
PKM P14618 1/20 0.52
TP53 P04637 1/20 0.51
ALOX15 P16050 1/20 0.51
ABCB1 P08183 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.51
CCR5 P51681 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22017772 0.84 BRAF (0.64) EGFR
SCHEMBL12345537 0.83 NPC1 (0.62) KMT2ALMNAALDH1A1HPGDSMN1; SMN2
SCHEMBL13880941 0.82 KMT2A (0.58) KMT2AEGFRLMNAALDH1A1HPGD
SCHEMBL2217357 0.81 HDAC8 (0.64) KMT2AALDH1A1HPGDSMN1; SMN2USP2
SCHEMBL2215952 0.80 HDAC8 (0.63) KMT2AALDH1A1SMN1; SMN2MAPTNPC1
SCHEMBL28668646 0.79 PKM (0.79) KMT2ALMNASMN1; SMN2MAPTHSD17B10
SCHEMBL15381993 0.79 ALDH1A1 (0.64) KMT2AEGFRLMNAALDH1A1HPGD
SCHEMBL22017395 0.78 EGFR (0.49) EGFRSMN1; SMN2MAPTHSD17B10WNT3A
SCHEMBL14845834 0.77 BTK (0.67) LMNAALDH1A1SMN1; SMN2MAPTNPC1
SCHEMBL21382964 0.77 RAB9A (0.60) EGFRLMNAALDH1A1MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098710-A1 SUBSTITUTED BIS-ARYL AMIDE COMPOUND AND PREPARATION METHOD AND APPLICATION THEREFOR 中国医学科学院医药生物技术研究所 2020-05-22 WO disclosed