SCHEMBL13891759

SCHEMBL13891759

Cc1cc(F)ccc1-c1nc(S(C)(=O)=O)nc2c1C(=O)N(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)CCCO2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.37
WDR5 P61964 5/20 0.35
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
TNIK Q9UKE5 2/20 0.33
TACR3 P29371 1/20 0.33
GRIN1 Q05586 2/20 0.32
GRIN2B Q13224 2/20 0.32
ADRB2 P07550 1/20 0.32
FPR1 P21462 1/20 0.32
GPR183 P32249 1/20 0.32
APLNR P35414 1/20 0.32
GLP1R P43220 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
GPR35 Q9HC97 1/20 0.32
P2RX7 Q99572 2/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891738 0.89 TACR1 (0.41) TACR1ROCK2ROCK1TNIKGRIN1
SCHEMBL13891737 0.87 TACR1 (0.41) TACR1WDR5ROCK2ROCK1TNIK
SCHEMBL13891616 0.85 SDHB (0.40) TACR1ROCK2ROCK1TNIKADRB2
SCHEMBL13891702 0.85 KDM4E (0.41) TACR1ROCK2ROCK1ADRB2FPR1
SCHEMBL13891740 0.79 TLR7 (0.36) P2RX7
SCHEMBL13891760 0.77 TACR1 (0.41) TACR1ROCK2ROCK1GRIN1GRIN2B
SCHEMBL13891705 0.77 MTOR (0.38) TACR1ROCK2ROCK1TNIKADRB2
SCHEMBL5232743 0.76 TACR1 (0.40) TACR1ADRB2FPR1GPR183APLNR
SCHEMBL5225462 0.75 SDHB (0.40) TACR1ADRB2FPR1GPR183APLNR
SCHEMBL13891719 0.74 TACR1 (0.48) TACR1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed