Olpadronic Acid

Olpadronic Acid

SCHEMBL138988

CN(C)CCC(O)(P(=O)(O)O)P(=O)(O)O

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FDPS P14324 20/20 0.58
GGPS1 O95749 8/20 0.58
PDE3A Q14432 3/20 0.58
AGTR1 P30556 1/20 0.58
OPRM1 P35372 1/20 0.58
LMNA P02545 1/20 0.50
ADRB3 P13945 1/20 0.50
PDE4D Q08499 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Olpadronic Acid SCHEMBL232124 0.98 FDPS (0.56) FDPSGGPS1PDE3AAGTR1OPRM1
Olpadronic Acid SCHEMBL9581942 0.90 FDPS (0.69) FDPSGGPS1PDE3AAGTR1OPRM1
SCHEMBL12631211 0.89 FDPS (0.49) FDPSGGPS1PDE3AAGTR1OPRM1
Olpadronic Acid SCHEMBL7457593 0.87 FDPS (0.71) FDPSGGPS1PDE3AAGTR1OPRM1
SCHEMBL3976360 0.86 FDPS (0.57) FDPSGGPS1PDE3AAGTR1OPRM1
Olpadronic Acid SCHEMBL5717996 0.86 FDPS (0.55) FDPSGGPS1PDE3AAGTR1OPRM1
SCHEMBL9333595 0.85 FDPS (0.61) FDPSGGPS1PDE3AAGTR1OPRM1
SCHEMBL8050318 0.84 FDPS (0.45) FDPSGGPS1PDE3AAGTR1OPRM1
SCHEMBL16091938 0.83 FDPS (0.62) FDPSGGPS1PDE3AAGTR1OPRM1
SCHEMBL9333367 0.83 FDPS (0.62) FDPSGGPS1PDE3AAGTR1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2429 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260102414-A1 USE OF DERIVATIVES CONTAINING C-O-P BONDS IN PATIENTS WITH KIDNEY FAILURE SANIFIT THERAPEUTICS S A (ES) 2026-04-16 US claimed
US-12569507-B2 CAR T-cells for the treatment of bone metastatic cancer H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2026-03-10 US claimed
EP-4684811-A1 NOVEL TREATMENT REGIMEN AND METHODS IN BONE HEALING Moroxite AB (SE) 2026-01-28 EP claimed
WO-2025261951-A1 COMBINATION THERAPY WITH AN ANTI-CA19-9 ANTIBODY AND FOLFIRINOX IN THE TREATMENT OF CANCER BioNTech SE (DE) 2025-12-26 WO claimed
US-20250295676-A1 INOSITOL PHOSPHATE COMPOUNDS FOR USE IN TREATING, INHIBITING THE PROGRESSION, OR PREVENTING CARDIOVASCULAR CALCIFICATION VIFOR (INTERNATIONAL) LTD. (CH) 2025-09-25 US claimed
EP-4611104-A1 NON-AQUEOUS ELECTROLYTE, SODIUM-ION BATTERY CONTAINING SAME, AND ELECTRICAL APPARATUS Contemporary Amperex Technology (Hong Kong) Limited (HK) 2025-09-03 EP claimed
EP-3901283-B1 THERAPEUTIC TREATMENT OF BREAST CANCER BASED ON C-MAF STATUS INBIOMOTION SL (ES) 2025-08-06 EP claimed
US-12359191-B2 Polyanionic acids to improve recovery and minimize system loss WATERS TECHNOLOGIES CORPORATION (US) 2025-07-15 US claimed
US-20250219149-A1 NON-AQUEOUS ELECTROLYTE AND SODIUM-ION BATTERY AND ELECTRIC APPARATUS INCLUDING SUCH ELECTROLYTE CONTEMPORARY AMPEREX TECHNOLOGY (HONG KONG) LIMITED (CN) 2025-07-03 US claimed
CN-119656381-B Active organic-inorganic composite implant material and preparation method and application thereof 广东粤港澳大湾区黄埔材料研究院 2025-06-13 CN claimed
US-5358941-A Treatment of bone disorders, osteoporosis MERCK & CO., INC. (US) 1994-10-25 US claimed
WO-1994012200-A1 DRY MIX FORMULATION FOR BISPHOSPHONIC ACIDS MERCK & CO., INC. (US) 1994-06-09 WO claimed
EP-0600834-A1 Use of methanebisphosphonic acid derivatives for the manufacture of a medicament for fracture healing CIBA-GEIGY AG (CH) 1994-06-08 EP claimed
US-5296475-A Methanediphosphonic acids and crown compounds for treatment of bone disorders or hypercalcemia CIBA-GEIGY CORPORATION (US) 1994-03-22 US claimed
WO-1994000129-A1 USE OF PHOSPHONATES FOR THE TREATMENT OF OSTEOPOROSIS PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1994-01-06 WO claimed
EP-0550385-A1 Oral pharmaceutical compositions containing derivatives of methane-diphosphonic acid and 18-crown-6 ethers CIBA-GEIGY AG (CH) 1993-07-07 EP claimed
US-5139786-A Topical formulations CIBA-GEIGY CORPORATION (US) 1992-08-18 US claimed
EP-0407345-A2 Topical formulations CIBA-GEIGY AG (CH) 1991-01-09 EP claimed
EP-0401243-A1 MEDICINAL PREPARATIONS CHARACTERIZED BY A COMBINATION OF CYTOSTATIC AGENTS, HORMONAL THERAPEUTIC AGENTS AND PHOSPHONE DERIVATIVES. HENKEL KGAA (DE) 1990-12-12 EP claimed
WO-1989007453-A1 MEDICINAL PREPARATIONS CHARACTERIZED BY A COMBINATION OF CYTOSTATIC AGENTS, HORMONAL THERAPEUTIC AGENTS AND PHOSPHONE DERIVATIVES HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1989-08-24 WO claimed