SCHEMBL13908151

SCHEMBL13908151

CCCc1nc2cc(C(C)=O)ccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
KMT2A Q03164 1/20 0.47
HTT P42858 1/20 0.45
APEX1 P27695 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 1/20 0.43
CHRM1 P11229 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11203298 0.88 DDAH1 (0.51) KDM4EKMT2AHTTAPEX1NPC1
Hydrochloric Acid SCHEMBL8829839 0.86 HTR1A (0.49) KDM4EKMT2AHTTAPEX1NPC1
SCHEMBL8906504 0.85 L3MBTL1 (0.54) KDM4EKMT2AHTTNPC1RAB9A
SCHEMBL7996355 0.83 SMN1; SMN2 (0.51) KDM4EHTTRAB9AALDH1A1SMN1; SMN2
SCHEMBL15223716 0.82 HTT (0.40) KMT2AHTTAPEX1NPC1RAB9A
SCHEMBL27639305 0.81 F10 (0.57)
SCHEMBL8788713 0.80 APEX1 (0.56) KMT2AAPEX1NPC1RAB9AALDH1A1
SCHEMBL6368877 0.79 GAA (0.57) KDM4EKMT2ANPC1RAB9AALDH1A1
SCHEMBL11887806 0.78 APEX1 (0.64) KDM4EKMT2AAPEX1NPC1RAB9A
SCHEMBL7334277 0.78 APEX1 (0.53) APEX1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed