SCHEMBL13952129

SCHEMBL13952129

O=C1c2ccccc2C(=O)N1Cc1cccc(F)c1F

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.47
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
ACHE P22303 7/20 0.47
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
RECQL P46063 1/20 0.46
RPS6KA2 Q15349 1/20 0.45
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44
CA12 O43570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679487 0.87 ACHE (0.57) CASP3ACHECA12
SCHEMBL29819864 0.87 ACHE (0.57) CASP3ACHECA12
SCHEMBL3131037 0.83 RECQL (0.47) CASP3ACHEKDM4EGAARECQL
SCHEMBL18954708 0.83 ALDH1A1 (0.59) ACHETSHRCA12
SCHEMBL13442859 0.81 CASP3 (0.62) CASP3ACHECA12
SCHEMBL18668991 0.81 MEN1 (0.50) CASP3KDM4EGAARECQLRPS6KA2
SCHEMBL18668934 0.80 CA12 (0.55) CASP3RPS6KA2POLBTSHRCA12
SCHEMBL3089984 0.80 GAA (0.64) ACHEKDM4EGAARECQLTSHR
SCHEMBL28737150 0.79 KDM4E (0.63) KDM4EGAARECQLCA12
SCHEMBL20256749 0.79 CA12 (0.44) CASP3ACHEKDM4EGAARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026248-A2 HYDRAZIDE, AMIDE, PHTHALIMIDE AND PHTHALHYDRAZIDE ANALOGS AS INHIBITORS OF RETROVIRAL INTEGRASE THE GOVERNMENT OF THE UNITED STATES, AS REPRESENTED BY THE SECRETARY OF HEALTH AND HUMAN SERVICES, NATIONAL INSTITUTES OF HEALTH, OFFICE OF TECHNOLOGY TRANSFER (US) 2009-02-26 WO disclosed