SCHEMBL1396563

SCHEMBL1396563

CCOP(=O)(CS(=O)(=O)c1ccccc1)OCC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.53
ALDH1A1 P00352 2/20 0.48
LMNA P02545 2/20 0.48
KDM4E B2RXH2 1/20 0.48
NPSR1 Q6W5P4 1/20 0.44
HSD11B1 P28845 3/20 0.43
KCNH2 Q12809 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
POLB P06746 2/20 0.41
ACHE P22303 1/20 0.41
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
NR1I2 O75469 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1374250 0.84 ALDH1A1 (0.47) ALDH1A1LMNACA12CA1CA2
SCHEMBL30727315 0.83 LMNA (0.49) PSIP1ALDH1A1LMNAKDM4ENPSR1
SCHEMBL31248447 0.83 CA12 (0.44) ALDH1A1KDM4ECA12CA1CA2
SCHEMBL30811026 0.83 CA12 (0.44) ALDH1A1LMNAKDM4ECA12CA1
SCHEMBL23732506 0.83 GAA (0.55) PSIP1ALDH1A1LMNACA12CA1
SCHEMBL23919240 0.83 KMT2A (0.51) LMNACA12CA1CA2CA4
SCHEMBL7886274 0.83 PSIP1 (0.50) PSIP1ALDH1A1LMNAKDM4ENPSR1
SCHEMBL8942619 0.83 PSIP1 (0.50) PSIP1ALDH1A1LMNAKDM4ENPSR1
SCHEMBL30811038 0.83 PLCG1 (0.48) LMNANPSR1CA12CA1CA2
SCHEMBL7371896 0.82 GAA (0.56) ALDH1A1LMNAKDM4ECA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115029833-A Flame-retardant fancy yarn and preparation process thereof 江阴市聚鑫花式线有限公司 2022-09-09 CN claimed
CN-115012086-A Fancy yarn dyed by vegetable dye and processing technology thereof 江阴市聚鑫花式线有限公司 2022-09-06 CN claimed
EP-0839155-A1 CYSTEINE PROTEASE INHIBITORS FOR USE IN TREATMENT OF IgE MEDIATED ALLERGIC DISEASES PEPTIDE THERAPEUTICS LIMITED (GB) 1998-05-06 EP claimed
WO-1997004004-A1 CYSTEINE PROTEASE INHIBITORS FOR USE IN TREATMENT OF IgE MEDIATED ALLERGIC DISEASES PEPTIDE THERAPEUTICS LIMITED (GB) 1997-02-06 WO claimed
US-12491252-B2 Substituted 3-amino-5-phenylbenzamide compounds as covalent inhibitors of enhancer zeste homolog 2 (EZH2) and proteolysis-targeting chimeric derivatives thereof (PROTACs) that induce degradation of EZH2 NORTHWESTERN UNIVERSITY (US) 2025-12-09 US disclosed
CN-114805322-B Prins reaction and intermediate for synthesizing halichondrin macrolides and analogues thereof 卫材R&D管理有限公司 2025-05-30 CN disclosed
US-20240335546-A1 SUBSTITUTED 3-AMINO-5-PHENYLBENZAMIDE COMPOUNDS AS COVALENT INHIBITORS OF ENHANCER ZESTE HOMOLOG 2 (EZH2) AND PROTEOLYSIS-TARGETING CHIMERIC DERIVATIVES THEREOF (PROTACS) THAT INDUCE DEGRADATION OF EZH2 NORTHWESTERN UNIVERSITY 2024-10-10 US disclosed
US-20240262832-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2024-08-08 US disclosed
US-12042543-B2 Substituted 3-amino-5-phenylbenzamide compounds as covalent inhibitors of enhancer zeste homolog 2 (EZH2) and proteolysis-targeting chimeric derivatives thereof (PROTACs) that induce degradation of EZH2 NORTHWESTERN UNIVERSITY (US) 2024-07-23 US disclosed
US-20240180158-A1 COMPOUNDS HAVING SELECTIVE INACTIVATION ACTIVITY UNIVERSITY OF NORTH CAROLINA AT WILMINGTON (US) 2024-06-06 US disclosed
EP-4329881-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-03-06 EP disclosed
US-20230346953-A1 SUBSTITUTED 3-AMINO-5-PHENYLBENZAMIDE COMPOUNDS AS COVALENT INHIBITORS OF ENHANCER ZESTE HOMOLOG 2 (EZH2) AND PROTEOLYSIS-TARGETING CHIMERIC DERIVATIVES THEREOF (PROTACS) THAT INDUCE DEGRADATION OF EZH2 UNITED STATES GOVERNMENT 2023-11-02 US disclosed
WO-1996030353-A1 REVERSIBLE PROTEASE INHIBITORS ARRIS PHARMACEUTICAL CORPORATION (US) 1996-10-03 WO disclosed
US-5519048-A 3-(indol-3-yl)-propenoic acid derivatives and pharmaceutical compositions thereof MERRELL PHARMACEUTICALS INC. (US) 1996-05-21 US disclosed
EP-0701551-A1 3-(INDOL-3-YL) PROPENOIC ACID DERIVATIVES AND AS NMDA ANTAGONISTS MERRELL PHARMA INC (US) 1996-03-20 EP disclosed
WO-1995023222-A1 IRREVERSIBLE CYSTEINE PROTEASE INHIBITORS CONTAINING VINYL GROUPS CONJUGATED TO ELECTRON WITHDRAWING GROUPS KHEPRI PHARMACEUTICALS, INC. (US) 1995-08-31 WO disclosed
WO-1994027964-A1 3-(INDOL-3-YL) PROPENOIC ACID DERIVATIVES AND AS NMDA ANTAGONISTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-12-08 WO disclosed
EP-0063489-B1 4\"-MODIFIED METHYLENE OLEANDOMYCINS PFIZER INC. (US) 1984-06-27 EP disclosed
EP-0063489-A1 4\"-Modified methylene oleandomycins PFIZER INC. (US) 1982-10-27 EP disclosed
US-4336368-A 4 Deoxy-4-methylene oleandomycin and derivatives thereof PFIZER INC. (US) 1982-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240180158-A1 COMPOUNDS HAVING SELECTIVE INACTIVATION ACTIVITY GAA, MGAM, GBA3 PSIP1 4068/4885ALDH1A1 171/4885LMNA 3292/4885
US-12042543-B2 Substituted 3-amino-5-phenylbenzamide compounds as covalent inhibitors of enhancer zeste homolog 2 (EZH2) and proteolysis-targeting chimeric derivatives thereof (PROTACs) that induce degradation of EZH2 EZH2, BAZ2A, BAZ2B PSIP1 1270/4885ALDH1A1 2801/4885LMNA 2665/4885
US-20240262832-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF GBA1, GAA, GBA2 PSIP1 3786/4885ALDH1A1 1938/4885LMNA 2954/4885
US-20230346953-A1 SUBSTITUTED 3-AMINO-5-PHENYLBENZAMIDE COMPOUNDS AS COVALENT INHIBITORS OF ENHANCER ZESTE HOMOLOG 2 (EZH2) AND PROTEOLYSIS-TARGETING CHIMERIC DERIVATIVES THEREOF (PROTACS) THAT INDUCE DEGRADATION OF EZH2 EZH2, BAZ2A, BAZ2B PSIP1 1270/4885ALDH1A1 2801/4885LMNA 2665/4885
US-12491252-B2 Substituted 3-amino-5-phenylbenzamide compounds as covalent inhibitors of enhancer zeste homolog 2 (EZH2) and proteolysis-targeting chimeric derivatives thereof (PROTACs) that induce degradation of EZH2 EZH2, BAZ2A, BAZ2B PSIP1 1270/4885ALDH1A1 2801/4885LMNA 2665/4885
US-20240335546-A1 SUBSTITUTED 3-AMINO-5-PHENYLBENZAMIDE COMPOUNDS AS COVALENT INHIBITORS OF ENHANCER ZESTE HOMOLOG 2 (EZH2) AND PROTEOLYSIS-TARGETING CHIMERIC DERIVATIVES THEREOF (PROTACS) THAT INDUCE DEGRADATION OF EZH2 EZH2, BAZ2A, BAZ2B PSIP1 1270/4885ALDH1A1 2801/4885LMNA 2665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.