SCHEMBL1397657

SCHEMBL1397657

CC1(C)CCc2sc(CN(CCc3ccc(Cl)c(Cl)c3)C(=O)c3c(F)c(Cl)cc4cc[nH]c34)cc2C1

nearest known ligand 0.30

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 2/20 0.30
SIGMAR1 Q99720 2/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1397708 0.93
SCHEMBL1397700 0.89 MCL1 (0.31)
SCHEMBL1397672 0.87 EEF2K (0.30)
SCHEMBL1397699 0.82 C5AR1 (0.31)
SCHEMBL1397377 0.81 C5AR1 (0.31)
SCHEMBL1397670 0.77 ALDH1A1 (0.31) MEN1ALDH1A1TP53CYP1A2CYP2C19
SCHEMBL1397763 0.76 C5AR1 (0.32)
SCHEMBL1385947 0.76 ESRRG (0.36) CENPESIGMAR1MEN1ALDH1A1TP53
SCHEMBL1397397 0.74 C5AR1 (0.31)
SCHEMBL1397368 0.74 SIGMAR1 (0.31) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007726-B1 BENZAMIDE AND HETEROARENE DERIVATIVES AS CETP INHIBITORS HOFFMANN LA ROCHE (CH) 2011-03-02 EP disclosed