SCHEMBL1397684

SCHEMBL1397684

CC(C)(C)c1ccc(CN(CCc2cccc(C(F)(F)F)c2)C(=O)c2c(F)c(Cl)cc3cc[nH]c23)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 6/20 0.37
CDK8 P49336 2/20 0.36
SLC2A1 P11166 1/20 0.36
MGLL Q99685 1/20 0.35
CCR9 P51686 1/20 0.34
CETP P11597 1/20 0.34
CHRM5 P08912 1/20 0.34
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HDAC8 Q9BY41 2/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1386968 0.89 MEN1 (0.37) TRPM8SLC2A1MGLLMEN1LMNA
SCHEMBL1397545 0.89 CCR9 (0.34) CCR9MEN1CYP1A2CYP2C19KMT2A
SCHEMBL1397829 0.88 CCR9 (0.36) SLC2A1CCR9FLT3
SCHEMBL20768023 0.87 SLC2A1 (0.38) TRPM8CDK8SLC2A1MGLLMEN1
SCHEMBL1397553 0.86 TRPM8 (0.35) TRPM8CDK8SLC2A1MGLLMEN1
SCHEMBL1397688 0.86 TRPM8 (0.34) TRPM8CDK8SLC2A1MGLLCETP
SCHEMBL1386856 0.83 PPARG (0.35) SLC2A1MGLLCETPLMNAHDAC8
SCHEMBL1397717 0.82 MCL1 (0.34) CDK8SLC2A1MGLLMEN1LMNA
SCHEMBL1397658 0.80 TRPM8 (0.37) TRPM8SLC2A1CCR9CETPHDAC8
SCHEMBL1386237 0.79 ESRRG (0.34) TRPM8HDAC8HDAC11HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007726-B1 BENZAMIDE AND HETEROARENE DERIVATIVES AS CETP INHIBITORS HOFFMANN LA ROCHE (CH) 2011-03-02 EP disclosed