SCHEMBL1399265

SCHEMBL1399265

COc1ccc2[nH]cc(Sc3ccc(F)cc3CCN)c2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.60
HTR1A P08908 5/20 0.60
HTR1B P28222 3/20 0.60
TRPM8 Q7Z2W7 2/20 0.60
HTR1D P28221 2/20 0.60
CYP1A2 P05177 1/20 0.60
MAPT P10636 1/20 0.60
TSHR P16473 1/20 0.60
NFKB1 P19838 1/20 0.60
HTR2C P28335 1/20 0.60
HTR7 P34969 1/20 0.60
HTR6 P50406 1/20 0.60
HTR4 Q13639 1/20 0.60
BLM P54132 1/20 0.59
PMP22 Q01453 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
IDO1 P14902 3/20 0.56
TUBB4A P04350 3/20 0.52
TUBB P07437 3/20 0.52
TUBA3C P0DPH7 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4632750 0.91 HTR2A (0.60) HTR2AHTR1AHTR1BTRPM8HTR1D
SCHEMBL1399411 0.88 MPO (0.65) HTR2AHTR1ATRPM8TSHRIDO1
SCHEMBL1399238 0.87 HTR2A (0.60) HTR2AHTR1AHTR1BTRPM8HTR1D
SCHEMBL4632929 0.86 IDO1 (0.55) HTR2AHTR1AHTR1BTRPM8HTR1D
SCHEMBL1399200 0.85 HTR1A (0.64) HTR2AHTR1AHTR1BTRPM8HTR1D
SCHEMBL1399440 0.85 HTR2A (0.58) HTR2AHTR1ATRPM8HTR1DIDO1
SCHEMBL1399264 0.84 IDO1 (0.56) HTR2AHTR1AMAPTHTR4IDO1
SCHEMBL1399398 0.83 HTR2A (0.58) HTR2AHTR1ATRPM8IDO1TUBB4A
SCHEMBL1399448 0.83 HTR2A (0.58) HTR2AHTR1ATRPM8IDO1TUBB4A
SCHEMBL4632232 0.81 HTR2A (0.65) HTR2AHTR1ATRPM8HTR2CIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1860100-B1 2-(1H-indolylsulfanyl)-benzyl amine derivatives as SSRI LUNDBECK & CO AS H (DK) 2011-03-02 EP claimed