SCHEMBL14005199

SCHEMBL14005199

O=C(NCc1ccccc1)c1ccc(C(=O)N(CCCNc2ncccn2)N2CCOCC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
CNR2 P34972 1/20 0.42
MAPK1 P28482 2/20 0.41
HPGDS O60760 2/20 0.41
HTT P42858 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
POLB P06746 1/20 0.41
GRIN2B Q13224 1/20 0.41
ROCK2 O75116 2/20 0.40
ROCK1 Q13464 2/20 0.40
RPS6KA5 O75582 1/20 0.40
MAP4K4 O95819 1/20 0.40
PRKCG P05129 1/20 0.40
PRKACA P17612 1/20 0.40
RPS6KB1 P23443 1/20 0.40
AKT1 P31749 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14070629 0.77 ALDH1A1 (0.45) ALDH1A1CNR2MAPK1HTTLMNA
SCHEMBL14070632 0.73 ALDH1A1 (0.41) ALDH1A1CNR2MAPK1HTTLMNA
SCHEMBL14005185 0.72 TSHR (0.57) ALDH1A1MAPK1HTTMAPTPOLB
SCHEMBL4889055 0.69 ALDH1A1 (0.49) ALDH1A1CNR2HTTPOLBNAMPT
SCHEMBL4898157 0.69 ALDH1A1 (0.50) ALDH1A1CNR2MAPK1HTTMAPT
SCHEMBL14070483 0.69 ALDH1A1 (0.70) ALDH1A1CNR2MAPK1HTTLMNA
SCHEMBL12655383 0.66 EPHX2 (0.61) ALDH1A1GRIN2BCLK4HPGD
SCHEMBL4748286 0.66 ALDH1A1 (0.46) ALDH1A1CNR2HTTAKT1NAMPT
SCHEMBL11900090 0.65 HDAC6 (0.85) MAPK1LMNAPOLBROCK2ROCK1
SCHEMBL27815577 0.64 MMP13 (0.51) ALDH1A1MAPK1HPGDSHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080293711-A1 Chemokine receptor modulators METASTATIX, INC. 2008-11-27 US disclosed
US-20080293711-A1 Chemokine receptor modulators METASTATIX, INC. 2008-11-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080293711-A1 Chemokine receptor modulators CCR5, CCL2, CXCR4 ALDH1A1 1359/4885CNR2 496/4885MAPK1 587/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.