SCHEMBL14014665

SCHEMBL14014665

FC(F)(F)c1ccc(Cl)c(COc2ccc(-c3cnc4c(-c5nnn[nH]5)cnn4c3C3CCCCC3)cc2)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.33
FFAR4 Q5NUL3 1/20 0.33
GPR119 Q8TDV5 4/20 0.33
NR1H2 P55055 1/20 0.32
PRMT5 O14744 1/20 0.32
PLAT P00750 2/20 0.31
ALOX5 P09917 2/20 0.31
ABL1 P00519 2/20 0.31
NTRK1 P04629 2/20 0.31
LCK P06239 2/20 0.31
FYN P06241 2/20 0.31
CSF1R P07333 2/20 0.31
FLT1 P17948 2/20 0.31
FLT3 P36888 2/20 0.31
NEK2 P51955 2/20 0.31
TYRO3 Q06418 2/20 0.31
NTRK3 Q16288 2/20 0.31
NTRK2 Q16620 2/20 0.31
AURKB Q96GD4 2/20 0.31
PLK4 O00444 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14014630 0.92 GPR119 (0.34) ALOX5APFFAR4GPR119PRMT5PLAT
SCHEMBL14014669 0.87 S1PR1 (0.35) ALOX5APPRMT5JAK2JAK3
SCHEMBL4710343 0.86 CYP3A4 (0.39) ALOX5APFFAR4GPR119TYRO3AXL
SCHEMBL14014641 0.85 GABBR2 (0.37) GPR119PLATTYRO3AXLGABBR2
SCHEMBL14014668 0.84 S1PR1 (0.36) PDGFRA
SCHEMBL14014625 0.84 GPR119 (0.37) ALOX5APFFAR4GPR119PRMT5TYRO3
SCHEMBL14014662 0.82 SCN1A (0.36) ALOX5APPLATGABBR2GABBR1
SCHEMBL14014558 0.82 TNK2 (0.41) GPR119PLATABL1NTRK1LCK
Tetrazole SCHEMBL4710754 0.82 CYP3A4 (0.36) ALOX5APGPR119TYRO3AXLPDGFRA
SCHEMBL14014628 0.81 PDE2A (0.33) ALOX5APGPR119PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7449488-B2 Pyrazolopyrimidines as protein kinase inhibitors SCHERING CORPORATION (US) 2008-11-11 US disclosed
US-7449488-B2 Pyrazolopyrimidines as protein kinase inhibitors SCHERING CORPORATION (US) 2008-11-11 US disclosed
US-7196111-B2 Pyrazolo[1,5a]pyrimidine compounds as antiviral agents SCHERING CORPORATION (US) 2007-03-27 US disclosed
US-7196111-B2 Pyrazolo[1,5a]pyrimidine compounds as antiviral agents SCHERING CORPORATION (US) 2007-03-27 US disclosed