SCHEMBL14026564

SCHEMBL14026564

C(=C/n1cncn1)\c1cnc2c(c1)CCN2

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.40
NNMT P40261 2/20 0.39
ASIC3 Q9UHC3 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.32
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005277 0.72 NNMT (0.44) GRM5NNMTASIC3PIK3C3ALOX5AP
SCHEMBL29951191 0.70 NNMT (0.53) GRM5NNMTASIC3PIK3C3ALOX5AP
SCHEMBL14027114 0.70 GRM5 (0.39) GRM5NNMTASIC3
SCHEMBL4833036 0.68 PIK3CA (0.40)
SCHEMBL17173410 0.67 NNMT (0.49) NNMTPIK3C3
SCHEMBL13533931 0.67 AHR (0.41) GRM5NNMTASIC3ALOX5APFEN1
SCHEMBL17173454 0.66 KMT2A (0.49) GRM5NNMTPIK3C3
SCHEMBL620335 0.65 CHRNB2 (0.48) GRM5NNMTASIC3PIK3C3ALOX5AP
SCHEMBL8927087 0.64 CYP19A1 (0.41)
SCHEMBL8385495 0.63 ASIC3 (0.57) GRM5NNMTASIC3PIK3C3ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7446199-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-11-04 US disclosed