SCHEMBL14031886

SCHEMBL14031886

CNC(=O)c1[nH]nc2c1CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
ADORA1 P30542 2/20 0.41
ESR2 Q92731 1/20 0.39
NR1H2 P55055 2/20 0.39
F12 P00748 1/20 0.38
MAPT P10636 3/20 0.38
MTOR P42345 1/20 0.37
GRAMD1A Q96CP6 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 1/20 0.36
MKNK1 Q9BUB5 2/20 0.36
IGF1R P08069 1/20 0.35
GPR119 Q8TDV5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5070051 0.86 ADORA1 (0.49) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL13070458 0.81 ADORA1 (0.53) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL23794808 0.81 PARP1 (0.46) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL5069421 0.81 F12 (0.44) PARP1TNKS2PARP2ADORA1NR1H2
SCHEMBL22074889 0.80 PARP1 (0.45) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL22492346 0.80 ADORA1 (0.50) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL5070030 0.80 F12 (0.41) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL29386147 0.79 RBP4 (0.42) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL28700403 0.78 L3MBTL1 (0.41) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL23794846 0.78 PARP1 (0.44) PARP1TNKS2PARP2ADORA1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435820-B2 Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use AVENTIS PHARMA S.A. (FR) 2008-10-14 US disclosed