SCHEMBL14035489

SCHEMBL14035489

CCCCc1ccc2c(O)cc(-c3ccccc3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.56
PSMB5 P28074 1/20 0.48
TRPV1 Q8NER1 1/20 0.45
CTRC Q99895 1/20 0.43
EIF4A1 P60842 5/20 0.43
HSD11B1 P28845 1/20 0.42
TACR3 P29371 2/20 0.41
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14035529 0.85 DHODH (0.54) DHODHPSMB5TRPV1CTRCEIF4A1
SCHEMBL12708293 0.82 KDM4E (0.42) DHODHTACR3
SCHEMBL16229566 0.76 BCHE (0.43) DHODHPSMB5TACR3
SCHEMBL10155099 0.76 KDM4E (0.56)
SCHEMBL12201040 0.75 ESR1 (0.53) DHODH
SCHEMBL9705061 0.75 DHODH (0.52) DHODHPSMB5CTRCHSD11B1ADORA1
SCHEMBL14623967 0.75 KDM4E (0.55) TACR3ADORA1
SCHEMBL1256551 0.75 ACHE (0.61) DHODHTACR3
SCHEMBL16234057 0.74 DHODH (0.56) DHODHPSMB5TRPV1CTRCEIF4A1
SCHEMBL22827977 0.74 DHODH (0.56) DHODHPSMB5TRPV1CTRCEIF4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1505945-B1 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2008-11-05 EP disclosed