SCHEMBL14035529

SCHEMBL14035529

CCCCc1ccc2c(C)cc(-c3ccccc3)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.54
PSMB5 P28074 1/20 0.52
TRPV1 Q8NER1 1/20 0.46
HSD11B1 P28845 2/20 0.46
ALDH1A1 P00352 4/20 0.43
MAPT P10636 4/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
THRB P10828 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
TACR3 P29371 1/20 0.42
EIF4A1 P60842 2/20 0.42
CTRC Q99895 1/20 0.41
AHR P35869 1/20 0.41
KDM4E B2RXH2 2/20 0.41
RAB9A P51151 2/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14035489 0.85 DHODH (0.56) DHODHPSMB5TRPV1HSD11B1TACR3
SCHEMBL13541765 0.76 ALDH1A1 (0.55) PSMB5ALDH1A1MAPTMEN1KMT2A
SCHEMBL9705061 0.76 DHODH (0.52) DHODHPSMB5HSD11B1MAPTMEN1
SCHEMBL951744 0.76 MAPT (0.65) DHODHALDH1A1MAPTMEN1KMT2A
SCHEMBL24755295 0.76 HSD11B1 (0.59) DHODHPSMB5TRPV1HSD11B1ALDH1A1
SCHEMBL14319678 0.75 ALDH1A1 (0.50) PSMB5ALDH1A1MAPTMEN1KMT2A
SCHEMBL22827977 0.75 DHODH (0.56) DHODHPSMB5TRPV1HSD11B1ALDH1A1
SCHEMBL16234057 0.75 DHODH (0.56) DHODHPSMB5TRPV1HSD11B1ALDH1A1
SCHEMBL6859623 0.74 ALDH1A1 (0.63) DHODHALDH1A1MAPTMEN1KMT2A
SCHEMBL30946935 0.74 ALDH1A1 (0.63) DHODHALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1505945-B1 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2008-11-05 EP disclosed