SCHEMBL14044797

SCHEMBL14044797

CCc1ncc2cc(C(C)(C)C)ccc2n1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 7/20 0.37
KCNH2 Q12809 1/20 0.36
PDE10A Q9Y233 1/20 0.36
METAP2 P50579 1/20 0.35
LCK P06239 1/20 0.34
KIT P10721 1/20 0.34
SRC P12931 1/20 0.34
KDR P35968 1/20 0.34
KDM4E B2RXH2 1/20 0.33
CYP2D6 P10635 1/20 0.33
ALDH1A1 P00352 2/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ALOX5AP P20292 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24974559 0.78 ESR1 (0.34) PDE10AALDH1A1HPGDCYP1A2
Tert-Butylbenzene SCHEMBL27402238 0.78 TP53 (0.38) KDM4EALDH1A1CYP1A2
SCHEMBL18177013 0.77 SCN10A (0.39) SCN10AKCNH2PDE10AMETAP2LCK
SCHEMBL4548606 0.77 SCN10A (0.39) SCN10AKCNH2PDE10AMETAP2LCK
SCHEMBL13363088 0.77 CYP1A2 (0.46) KDM4EALDH1A1CYP1A2
SCHEMBL179533 0.76 LCK (0.52) SCN10AKCNH2LCKKITSRC
SCHEMBL13273390 0.76 HTR3A (0.48) PDE10AKDRKDM4EALDH1A1
SCHEMBL30781766 0.76 NOS1 (0.34)
SCHEMBL24204603 0.76 EGFR (0.49) KCNH2PDE10ALCKKDRKDM4E
SCHEMBL19104136 0.76 ALDH1A1 (0.42) SCN10AKCNH2PDE10AMETAP2LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435823-B2 Compounds and methods of use AMGEN INC. (US) 2008-10-14 US disclosed