SCHEMBL1406497

SCHEMBL1406497

CCOC(=O)c1cc2cc(Cl)c(O)c([N+](=O)[O-])c2oc1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.59
MAOB P27338 7/20 0.56
MAOA P21397 2/20 0.53
GPR35 Q9HC97 1/20 0.51
MIF P14174 1/20 0.47
PFKFB3 Q16875 1/20 0.47
KDM4E B2RXH2 5/20 0.44
HSD17B10 Q99714 2/20 0.44
ALDH1A1 P00352 3/20 0.43
GLA P06280 3/20 0.43
GAA P10253 3/20 0.43
CA12 O43570 2/20 0.43
CA2 P00918 2/20 0.43
CA3 P07451 2/20 0.43
CA4 P22748 2/20 0.43
CA6 P23280 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
CA14 Q9ULX7 2/20 0.43
HPGD P15428 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1406333 0.88 MAPT (0.60) MAPTMAOBMAOAGPR35MIF
SCHEMBL1406456 0.88 MAPT (0.60) MAPTMAOBMAOAGPR35MIF
SCHEMBL6478938 0.86 MAPT (0.70) MAPTMAOBMAOAGPR35MIF
SCHEMBL1406624 0.82 GPR35 (0.73) MAOBMAOAGPR35KDM4EHSD17B10
SCHEMBL1406713 0.81 MAPT (0.64) MAPTMAOBMAOAGPR35MIF
SCHEMBL6110097 0.81 MAPT (0.62) MAPTMAOBMAOAGPR35MIF
SCHEMBL1406246 0.80 MAPT (0.53) MAPTMAOBMAOAGPR35MIF
SCHEMBL6109314 0.80 MAPT (0.61) MAPTMAOBMAOAGPR35MIF
SCHEMBL1406806 0.76 MAPT (0.66) MAPTMAOBMAOAGPR35MIF
SCHEMBL11494991 0.76 MAOB (0.77) MAPTMAOBMAOAGPR35MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295053-B1 Novel 2H-chromen-2-one-3-carboxamides for medical uses INST MATERIA MEDICA CAMS (CN) 2016-10-19 EP disclosed
US-8338401-B2 Coumarin-amide derivatives and its preparation, said drug composition and its use INSTITUTE OF MATERIA MEDICA CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2012-12-25 US disclosed
US-8338401-B2 Coumarin-amide derivatives and its preparation, said drug composition and its use INSTITUTE OF MATERIA MEDICA CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2012-12-25 US disclosed
EP-2295053-A1 Novel 2H-chromen-2-one-3-carboxamides for medical uses THE INSTITUTE OF MATERIA MEDICA OF CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2011-03-16 EP disclosed
WO-2008013928-A2 TREATMENT OF CANCER WITH INTERFERON GENE DELIVERY IN COMBINATION WITH A TGF-BETA INHIBITOR BIOGEN IDEC MA INC. (US) 2008-01-31 WO disclosed
US-20060148834-A1 Novel coumarin-amide derivatives and its preparation, said drug composition and its use INSTITUTE OF MATERIA MEDICA CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2006-07-06 US disclosed
EP-1570846-A1 THE NOVEL COUMARIN-AMIDE DERIVATIVES AND ITS PREPARATION, SAID DRUG COMPOSITION AND ITS USE THE INSTITUTE OF MATERIA MEDICA OF CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2005-09-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060148834-A1 Novel coumarin-amide derivatives and its preparation, said drug composition and its use INSR, GLS, INSRR MAPT 3985/4885MAOB 4669/4885MAOA 4761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.