SCHEMBL14080975

SCHEMBL14080975

Nc1c(N2CCNCC2)cnn(-c2ccccc2)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.54
NPC1 O15118 5/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
LMNA P02545 2/20 0.51
POLB P06746 1/20 0.51
KMT2A Q03164 1/20 0.51
ALDH1A1 P00352 5/20 0.47
DCTPP1 Q9H773 2/20 0.47
MAPT P10636 4/20 0.46
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
ADRB1 P08588 1/20 0.46
HTR3A P46098 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
HTR1A P08908 1/20 0.45
HTR7 P34969 1/20 0.45
HTR2B P41595 1/20 0.45
HTR6 P50406 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13942534 0.87 NPC1 (0.70) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL13942543 0.86 NPC1 (0.71) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL6030180 0.84 ALDH1A1 (0.66) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL13942545 0.84 NPC1 (0.72) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL13304485 0.79 NPC1 (0.65) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL8237031 0.78 MAPT (0.51) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL17057998 0.77 NPC1 (0.50) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL14082616 0.77 HTR1A (0.52) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL17058099 0.77 RAB9A (0.50) RAB9ANPC1SMN1; SMN2LMNAPOLB
SCHEMBL14081526 0.77 ALDH1A1 (0.56) RAB9ANPC1SMN1; SMN2LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115385-A2 PIPERAZINE-SUBSTITUTED PYRIDAZINONE DERIVATIVES USEFUL AS GLUCAN SYNTHASE INHIBITORS SCHERING CORPORATION (US) 2008-09-25 WO disclosed
WO-2008115381-A1 PYRIDAZINONE DERIVATIVES USEFUL AS GLUCAN SYNTHASE INHIBITORS SCHERING CORPORATION (US) 2008-09-25 WO disclosed