SCHEMBL14090197

SCHEMBL14090197

C=CCOC(=O)N[C@H]1C[C@@H](C(=O)OC)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 11/20 0.38
CYP19A1 P11511 1/20 0.38
ANPEP P15144 6/20 0.36
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
KCNA3 P22001 1/20 0.33
PTPN1 P18031 1/20 0.33
BTK Q06187 1/20 0.33
ALDH1A1 P00352 1/20 0.33
P2RX3 P56373 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3894190 1.00 MMP2 (0.38) MMP2CYP19A1ANPEPNR1H2NR1H3
SCHEMBL29697301 0.90 BTK (0.39) MMP2ANPEPNR1H2KCNA3BTK
SCHEMBL3898037 0.90 BTK (0.39) MMP2ANPEPNR1H2KCNA3BTK
SCHEMBL7727315 0.84 BTK (0.46) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL7727313 0.84 BTK (0.46) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL7731684 0.84 BTK (0.46) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL12480680 0.84 MMP2 (0.40) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL9907303 0.84 MMP2 (0.40) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL13938226 0.80 MMP2 (0.47) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL13938227 0.80 MMP2 (0.47) MMP2ANPEPNR1H2NR1H3PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12358886-B2 Heterocyclic compounds for use in the treatment of cancer ARTIOS PHARMA LIMITED (GB) 2025-07-15 US disclosed
CN-114667167-B Heterocyclic compounds for the treatment of cancer 阿提奥斯医药有限公司 2024-12-20 CN disclosed
EP-4010080-B1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LTD (GB) 2023-09-27 EP disclosed
US-20230242503-A9 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LIMITED (GB) 2023-08-03 US disclosed
US-20230242503-A9 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LIMITED (GB) 2023-08-03 US disclosed
US-20230242503-A9 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LIMITED (GB) 2023-08-03 US disclosed
US-20220298134-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LIMITED (GB) 2022-09-22 US disclosed
US-20220298134-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LIMITED (GB) 2022-09-22 US disclosed
CN-114667167-A Heterocyclic compounds for the treatment of cancer 阿提奥斯医药有限公司 2022-06-24 CN disclosed
EP-4010080-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER Artios Pharma Limited (GB) 2022-06-15 EP disclosed
WO-2021028643-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LIMITED (GB) 2021-02-18 WO disclosed
US-7417024-B2 Template-fixed peptidomimetics as inhibitors of serine proteases POLYPHOR LTD. (CH) 2008-08-26 US disclosed
US-7253146-B2 Template-fixed peptidomimetics with antimicrobial activity POLYPHOR LTD (CH) 2007-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242503-A9 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER SDHA, SDHB, NQO1 MMP2 1545/4885CYP19A1 19/4885ANPEP 1719/4885
US-20220298134-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER SDHA, SDHB, NQO1 MMP2 1545/4885CYP19A1 19/4885ANPEP 1719/4885
US-12358886-B2 Heterocyclic compounds for use in the treatment of cancer SDHA, DPYD, TP53 MMP2 2027/4885CYP19A1 75/4885ANPEP 1431/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.