Methandrostenolone

Methandrostenolone

SCHEMBL140928

C[C@]12C=CC(=O)C=C1CC[C@@H]1[C@@H]2CC[C@@]2(C)[C@H]1CC[C@]2(C)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

AR

The experimentally established mechanism targets of Methandrostenolone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 1.00
MAPT P10636 2/20 1.00
CYP19A1 P11511 9/20 0.65
CYP3A4 P08684 1/20 0.65
GUSB P08236 1/20 0.65
SHBG P04278 2/20 0.63
ALDH1A1 P00352 2/20 0.60
NR3C1 P04150 2/20 0.60
PGR P06401 2/20 0.60
ADRA1A P35348 1/20 0.60
HTR2B P41595 1/20 0.60
HSD17B10 Q99714 3/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
HIF1A Q16665 1/20 0.53
SLC29A1 Q99808 1/20 0.53
TDP1 Q9NUW8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methandrostenolone SCHEMBL28423591 1.00 LMNA (1.00) LMNAMAPTCYP19A1CYP3A4GUSB
Methandrostenolone SCHEMBL8408550 1.00 LMNA (1.00) LMNAMAPTCYP19A1CYP3A4GUSB
Methandrostenolone SCHEMBL21177905 1.00 LMNA (1.00) LMNAMAPTCYP19A1CYP3A4GUSB
Methandrostenolone SCHEMBL4435272 1.00 LMNA (1.00) LMNAMAPTCYP19A1CYP3A4GUSB
Methandrostenolone SCHEMBL16755284 1.00 LMNA (1.00) LMNAMAPTCYP19A1CYP3A4GUSB
Methandrostenolone SCHEMBL6395376 0.90 LMNA (0.81) LMNAMAPTCYP19A1CYP3A4GUSB
SCHEMBL5270893 0.90 LMNA (0.81) LMNAMAPTCYP19A1CYP3A4ALDH1A1
SCHEMBL10861103 0.90 LMNA (0.81) LMNAMAPTCYP19A1CYP3A4ALDH1A1
SCHEMBL17775770 0.87 LMNA (0.77) LMNAMAPTCYP19A1CYP3A4
SCHEMBL27046922 0.86 LMNA (0.75) LMNAMAPTCYP19A1CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3084 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119570811-A Vinca EIN3-EILs transcription factor and application thereof 上海交通大学 2025-03-07 CN claimed
CN-119202111-A Knowledge graph-based arch dam abutment unfavorable structural surface treatment measure recommendation method and terminal equipment 中国电建集团中南勘测设计研究院有限公司 2024-12-27 CN claimed
US-20240358719-A1 Formulations for Prolonging Gestation and for Complications of Menstruation or Gestation THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2024-10-31 US claimed
EP-3863708-B1 MIXED IONIC CONDUCTORS AND CORRESPONDING DEVICES, SYSTEMS AND METHODS OF MAKING BATTELLE MEMORIAL INSTITUTE (US) 2024-09-11 EP claimed
EP-3612223-B1 TREATING MALE SENESCENCE NAT INSTITUTE OF BIOLOGICAL SCIENCES BEIJING (CN) 2024-07-31 EP claimed
CN-118154052-A Power distribution network power exchange station site selection planning method considering centralized charging mode 国网湖北省电力有限公司电力科学研究院 2024-06-07 CN claimed
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
CN-117630146-A Nondestructive testing method for pollutants in aquatic products 北京市农产品质量安全中心 2024-03-01 CN claimed
EP-4313061-A1 FORMULATIONS FOR PROLONGING GESTATION AND FOR COMPLICATIONS OF MENSTRUATION OR GESTATION The Board of Trustees of the Leland Stanford Junior University (US) 2024-02-07 EP claimed
US-20230301931-A1 NANOPARTICULATE SYSTEM FOR TREATING ORAL CANCER THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2023-09-28 US claimed
EP-0240904-B1 PROCESS FOR THE PREPARATION OF SOLID PHARMACEUTICAL FORMS BASF Aktiengesellschaft (DE) 1992-07-01 EP claimed
US-5073379-A Melts, extrusion, rolling. tablets BASF AKTIENGESELLSCHAFT (DE) 1991-12-17 US claimed
US-5071657-A DEVICE FOR TRANSDERMAL ADMINISTRATION OF ACTIVE MEDICINAL AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 1991-12-10 US claimed
US-5026692-A Prevention and treatment of immunodeficiency diseases RESEARCH DEVELOPMENT CORPORATION OF JAPAN (JP) 1991-06-25 US claimed
EP-0199768-A4 A METHOD FOR THE PREVENTION OF OCULAR HYPERTENSION, TREATMENT OF GLAUCOMA AND TREATMENT OF OCULAR HYPERTENSION. KNEPPER PAUL A 1989-04-26 EP claimed
US-4801460-A N-VINYLPYRROLIDONE POLYMER BINDER BASF AKTIENGESELLSCHAFT (DE) 1989-01-31 US claimed
EP-0199768-A1 A METHOD FOR THE PREVENTION OF OCULAR HYPERTENSION, TREATMENT OF GLAUCOMA AND TREATMENT OF OCULAR HYPERTENSION KNEPPER, Paul A. (US) 1986-11-05 EP claimed
US-4617299-A ADMINISTERING SELECTED ANABOLIC ANDROGENIC COMPOUNDS KNEPPER PAUL A (US) 1986-10-14 US claimed
WO-1986002554-A1 A METHOD FOR THE PREVENTION OF OCULAR HYPERTENSION, TREATMENT OF GLAUCOMA AND TREATMENT OF OCULAR HYPERTENSION KNEPPER PAUL A 1986-05-09 WO claimed
US-4346709-A Drug delivery devices comprising erodible polymer and erosion rate modifier ALZA CORPORATION (US) 1982-08-31 US claimed