SCHEMBL14099345

SCHEMBL14099345

COc1cc(-c2cc3c(c(C(C)=O)c2)OCC3)cc(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
PARP1 P09874 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ERN1 O75460 2/20 0.38
PDE4A P27815 1/20 0.36
CYP2A6 P11509 1/20 0.34
PLK1 P53350 1/20 0.33
HTT P42858 1/20 0.33
KDM1A O60341 1/20 0.32
PIN1 Q13526 1/20 0.32
CREBBP Q92793 1/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
MAP2K1 Q02750 3/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640425 0.91 PARP1 (0.42) KDM4EPARP1ALDH1A1LMNAHSD17B10
SCHEMBL4640440 0.89 PARP1 (0.41) KDM4EPARP1ALDH1A1LMNAHSD17B10
SCHEMBL4640372 0.78 JAK2 (0.46) KDM4EPARP1ALDH1A1LMNAHSD17B10
SCHEMBL4642112 0.75 KDM4E (0.46) KDM4EPARP1ALDH1A1LMNAHSD17B10
SCHEMBL4640351 0.74 ALDH1A1 (0.49) KDM4EALDH1A1LMNAHSD17B10ERN1
SCHEMBL4740085 0.71 PARP1 (0.50) PARP1ERN1CYP2A6CREBBP
SCHEMBL5032923 0.69 PARP1 (0.49) KDM4EPARP1ALDH1A1LMNAHSD17B10
SCHEMBL3945829 0.68 KDM4E (0.45) KDM4EALDH1A1LMNAHSD17B10ERN1
SCHEMBL26462283 0.68 LMNA (0.50) KDM4EPARP1ALDH1A1LMNAHSD17B10
SCHEMBL219830 0.68 HTR3A (0.50) KDM4EPARP1ALDH1A1LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1956016-A1 Bicyclic acyltryptophanols Bayer Schering Pharma Aktiengesellschaft (DE) 2008-08-13 EP disclosed