SCHEMBL14101711

SCHEMBL14101711

Cc1ccccc1-c1nn(-c2cc(N3CCCC3)ccc2C(F)(F)F)c(=O)c2c1CCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.42
MAPK1 P28482 2/20 0.42
HTT P42858 2/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
NPSR1 Q6W5P4 3/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
P2RX7 Q99572 1/20 0.37
NOTUM Q6P988 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
HTR6 P50406 1/20 0.35
AR P10275 1/20 0.35
PDK2 Q15119 2/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720706 0.88 P2RX7 (0.42) NPSR1CYP3A4CYP2C9P2RX7PDK2
SCHEMBL4720711 0.88 P2RX7 (0.42) NPSR1CYP3A4CYP2C9P2RX7PDK2
SCHEMBL14101706 0.85 MAPT (0.38) MAPTMAPK1HTTALDH1A1POLB
SCHEMBL14101792 0.83 NOTUM (0.39) MAPTMAPK1HTTALDH1A1POLB
SCHEMBL14101882 0.82 KDM4E (0.39) MAPTMAPK1HTTALDH1A1POLB
SCHEMBL14101798 0.82 PDE4A (0.38) MAPTMAPK1HTTALDH1A1POLB
SCHEMBL14101794 0.82 PTGS2 (0.42) MAPTMAPK1HTTALDH1A1POLB
SCHEMBL14101783 0.82 NOTUM (0.38) MAPTMAPK1HTTALDH1A1POLB
SCHEMBL14101895 0.81 P2RX7 (0.38) MAPTMAPK1HTTALDH1A1POLB
SCHEMBL4724195 0.81 F10 (0.42) MAPTMAPK1HTTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed