SCHEMBL14101790

SCHEMBL14101790

O=C(O)c1ccc(-c2nn(-c3cc(N4CCCC4)ccc3C(F)(F)F)c(=O)c3c2CCC3)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.42
TTR P02766 2/20 0.38
PPARG P37231 1/20 0.37
RARA P10276 1/20 0.37
RARB P10826 1/20 0.37
RARG P13631 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
NOTUM Q6P988 2/20 0.36
CHEK1 O14757 1/20 0.36
FAAH O00519 1/20 0.35
NTRK1 P04629 1/20 0.35
IP6K1 Q92551 1/20 0.35
IP6K3 Q96PC2 1/20 0.35
IP6K2 Q9UHH9 1/20 0.35
ADH5 P11766 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723772 0.89 RORC (0.42) RORCTTRNOTUM
SCHEMBL4723777 0.89 RORC (0.42) RORCTTRNOTUM
SCHEMBL14101882 0.89 KDM4E (0.39) PDE4APDE4BPDE4CPDE4DNOTUM
SCHEMBL14101794 0.88 PTGS2 (0.42) PDE4APDE4BPDE4CPDE4DNOTUM
SCHEMBL14101706 0.84 MAPT (0.38) PDE4APDE4BPDE4CPDE4DNOTUM
SCHEMBL14101736 0.83 NOTUM (0.37) PDE4APDE4BPDE4CPDE4DNOTUM
SCHEMBL14101798 0.83 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DNOTUM
SCHEMBL4724195 0.81 F10 (0.42) PDE4APDE4BPDE4CPDE4DNOTUM
SCHEMBL14101895 0.81 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DNOTUM
SCHEMBL4720673 0.81 LCK (0.41) RORCPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed