SCHEMBL14101987

SCHEMBL14101987

COC(=O)CN1CCc2c(-c3ccc(F)c(C)c3)nn(-c3cc(F)ccc3C(F)(F)F)c(=O)c21

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 2/20 0.34
TP53 P04637 1/20 0.34
TRPM2 O94759 1/20 0.33
THRB P10828 1/20 0.33
GRIN2B Q13224 4/20 0.33
P2RX7 Q99572 3/20 0.33
MAPK14 Q16539 1/20 0.32
GRIN1 Q05586 1/20 0.32
DPP4 P27487 2/20 0.32
DPP8 Q6V1X1 2/20 0.32
AR P10275 1/20 0.32
DPP9 Q86TI2 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
C5AR1 P21730 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722057 0.91 GRIN2B (0.35) KCNK3THRBGRIN2BP2RX7GRIN1
SCHEMBL4720752 0.88 LGALS3 (0.34) KCNK3GRIN2BP2RX7CNR2
SCHEMBL14102047 0.82 AR (0.34) TRPM2AR
SCHEMBL4718895 0.76 CYP3A4 (0.32) C5AR1
SCHEMBL4722852 0.75 GRIN1 (0.34) KCNK3GRIN2BGRIN1
SCHEMBL4718914 0.75 P2RX7 (0.36) P2RX7
SCHEMBL4718912 0.75 P2RX7 (0.36) P2RX7
SCHEMBL4724182 0.75 P2RX7 (0.36) P2RX7
SCHEMBL4719091 0.74 F10 (0.36) P2RX7
SCHEMBL4719085 0.74 F10 (0.36) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed