SCHEMBL4722057

SCHEMBL4722057

Cc1cc(-c2nn(-c3cc(F)ccc3C(F)(F)F)c(=O)c3c2CCN3CC(=O)O)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 9/20 0.35
AKR1B1 P15121 2/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
AKR1B10 O60218 1/20 0.34
P2RX7 Q99572 3/20 0.33
KCNK3 O14649 2/20 0.33
THRB P10828 1/20 0.33
GRIN1 Q05586 1/20 0.33
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14101987 0.91 KCNK3 (0.34) GRIN2BP2RX7KCNK3THRBGRIN1
SCHEMBL4720752 0.90 LGALS3 (0.34) GRIN2BP2RX7KCNK3
SCHEMBL4722667 0.81 AR (0.34) AKR1B1AKR1B10P2RX7
SCHEMBL4718895 0.78 CYP3A4 (0.32)
SCHEMBL4720926 0.77 WDR5 (0.33) AKR1B1PTGDR2AKR1B10
SCHEMBL4722852 0.77 GRIN1 (0.34) GRIN2BKCNK3GRIN1
SCHEMBL4724182 0.77 P2RX7 (0.36) P2RX7
SCHEMBL4718912 0.77 P2RX7 (0.36) P2RX7
SCHEMBL4718914 0.77 P2RX7 (0.36) P2RX7
SCHEMBL14101709 0.75 F10 (0.39) AKR1B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed