SCHEMBL14130573

SCHEMBL14130573

Oc1ccc(NCl)c2cccnc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.64
KDM4E B2RXH2 11/20 0.61
HSP90AA1 P07900 3/20 0.61
LMNA P02545 2/20 0.61
MAPT P10636 2/20 0.61
BRD4 O60885 1/20 0.61
METAP2 P50579 1/20 0.61
METAP1 P53582 1/20 0.61
MMP2 P08253 4/20 0.56
L3MBTL1 Q9Y468 5/20 0.56
HTT P42858 3/20 0.56
MPI P34949 1/20 0.56
HSP90AB1 P08238 1/20 0.56
PSMB5 P28074 1/20 0.56
SLC6A2 P23975 1/20 0.56
NPC1 O15118 4/20 0.54
RAB9A P51151 3/20 0.54
GAA P10253 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
MMP9 P14780 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24081122 0.84 IDO1 (0.66) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL28942142 0.82 IDO1 (0.64) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL22705016 0.82 IDO1 (0.64) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL15217626 0.82 IDO1 (0.69) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL1920452 0.78 KDM4E (0.70) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL12599074 0.78 IDO1 (1.00) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL12599076 0.78 IDO1 (1.00) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL7032474 0.77 IDO1 (0.61) IDO1KDM4EHSP90AA1LMNAMAPT
SCHEMBL27816447 0.77 KDM4E (0.68) IDO1KDM4EHSP90AA1LMNAMAPT
Methane SCHEMBL27551425 0.77 KDM4E (0.68) IDO1KDM4EHSP90AA1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9302993-B2 8-hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2016-04-05 US disclosed
US-20150335635-A1 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LIMITED (AU) 2015-11-26 US disclosed
US-20150335635-A1 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LIMITED (AU) 2015-11-26 US disclosed
US-8975278-B2 8-hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2015-03-10 US disclosed
US-8975278-B2 8-hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2015-03-10 US disclosed
US-20080161353-A1 8-Hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2008-07-03 US disclosed
US-20080161353-A1 8-Hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2008-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150335635-A1 8-HYDROXY QUINOLINE DERIVATIVES PARK7, COQ8A, NLN IDO1 1644/4885KDM4E 3604/4885HSP90AA1 1187/4885
US-20080161353-A1 8-Hydroxy quinoline derivatives PARK7, COQ8A, NLN IDO1 1644/4885KDM4E 3604/4885HSP90AA1 1187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.