SCHEMBL14136285

SCHEMBL14136285

CCCN1CB(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.50
PNMT P11086 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
KDM2B Q8NHM5 1/20 0.39
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13698268 0.90 SIGMAR1 (0.52) SIGMAR1CYP1A2CYP2D6TMEM97DRD2
SCHEMBL13698294 0.86 SIGMAR1 (0.45) SIGMAR1PNMTCYP1A2CYP2D6TMEM97
SCHEMBL13698270 0.80 CYP2D6 (0.42) SIGMAR1CYP1A2CYP2D6TMEM97
SCHEMBL7528803 0.67 SIGMAR1 (1.00) SIGMAR1CYP1A2CYP2D6TMEM97TP53
SCHEMBL2922701 0.67 SIGMAR1 (0.62) SIGMAR1DRD2DRD3
SCHEMBL11938899 0.67 SIGMAR1 (0.77) SIGMAR1CYP1A2CYP2D6TMEM97
SCHEMBL13698300 0.66 RAB9A (0.36) DRD2DRD3
SCHEMBL13698247 0.64 DRD2 (0.60) SIGMAR1KDM2BDRD2DRD3
SCHEMBL3860327 0.63 DRD2 (0.57) SIGMAR1DRD2DRD3
SCHEMBL19261820 0.62 SIGMAR1 (0.48) SIGMAR1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8461196-B2 1-aryl-3-azabicyclo[3.1.0]hexanes: preparation and use to treat neuropsychiatric disorders DOV PHARMACEUTICAL 2013-06-11 US disclosed
US-20120302619-A1 Novel 1-aryl-3-Azabicyclo[3.1.0]Hexanes: Preparation And Use To Treat Neuropsychiatric Disorders OTSUKA AMERICA PHARMACEUTICAL, INC. 2012-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120302619-A1 Novel 1-aryl-3-Azabicyclo[3.1.0]Hexanes: Preparation And Use To Treat Neuropsychiatric Disorders HTR3C, HTR1B, HTR2C SIGMAR1 1402/4885PNMT 57/4885CYP1A2 188/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.