SCHEMBL14181753

SCHEMBL14181753

CC1(C)N/C(=C\C(=O)c2ccccc2)c2ccc(F)cc2O1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.36
PGR P06401 2/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
NPC1 O15118 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HPGD P15428 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
CCNB2 O95067 2/20 0.34
CDK1 P06493 2/20 0.34
CCNB1 P14635 2/20 0.34
CCNB3 Q8WWL7 2/20 0.34
TGM2 P21980 1/20 0.34
HSP90AA1 P07900 1/20 0.34
CCR6 P51684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4844537 0.91 PGR (0.38) RAB9APGRNPC1SMN1; SMN2HPGD
SCHEMBL4842742 0.87 RAB9A (0.38) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL4841185 0.86 TGM2 (0.37) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL4843983 0.85 RAB9A (0.41) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL4835742 0.84 TP53 (0.43) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL14181769 0.83 MAPT (0.39) RAB9ASMN1; SMN2TP53MAPTHSP90AA1
SCHEMBL4843746 0.80 RAB9A (0.38) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL14181858 0.79 RAB9A (0.39) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL4841022 0.79 CDYL2 (0.38) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL4835482 0.77 MAPT (0.43) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378428-B2 Nitrogen-containing bicyclic compounds and drugs containing the same as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-05-27 US disclosed