SCHEMBL14190849

SCHEMBL14190849

CC(=O)Nc1cccc(CN2CCC(N)CC2)c1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.55
MCHR2 Q969V1 1/20 0.55
MCHR1 Q99705 1/20 0.55
BTK Q06187 1/20 0.53
ACKR3 P25106 12/20 0.53
MEN1 O00255 1/20 0.52
TSHR P16473 1/20 0.52
KMT2A Q03164 1/20 0.52
CCR3 P51677 1/20 0.52
SMYD3 Q9H7B4 1/20 0.51
DCUN1D1 Q96GG9 1/20 0.51
SIRT1 Q96EB6 1/20 0.51
ACHE P22303 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4229523 0.91 SIRT1 (0.51) KCNH2MCHR2MCHR1BTKACKR3
SCHEMBL15933654 0.85 ACHE (0.58) KCNH2MCHR2MCHR1ACKR3CCR3
SCHEMBL10702311 0.85 KDM4E (0.67) BTKACKR3MEN1TSHRKMT2A
SCHEMBL16665723 0.84 ALDH1A1 (0.69) KCNH2MCHR1MEN1KMT2AACHE
SCHEMBL7600247 0.84 KDM4E (0.69) BTKACKR3MEN1TSHRKMT2A
SCHEMBL11000210 0.84 MEN1 (0.51) KCNH2MCHR2MCHR1BTKACKR3
Hydrochloric Acid SCHEMBL16654841 0.83 ALDH1A1 (0.68) KCNH2MCHR1MEN1KMT2AACHE
SCHEMBL17754101 0.82 SMN1; SMN2 (0.63) BTKACKR3MEN1TSHRKMT2A
SCHEMBL30577399 0.82 SMN1; SMN2 (0.63) BTKACKR3MEN1TSHRKMT2A
SCHEMBL11926135 0.82 CHRM3 (0.69) BTKMEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071587-A2 2-(PIPERIDIN-4-YL)-4-PHENOXY- OR PHENYLAMINO-PYRIMIDINE DERIVATIVES AS NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2008-06-19 WO disclosed