Sophoraflavanone A

Sophoraflavanone A

SCHEMBL141996

CC(C)=CCC/C(C)=C/Cc1c(O)cc(O)c2c1OC(c1ccc(O)cc1)CC2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 5/20 1.00
ESR1 P03372 7/20 0.83
ESR2 Q92731 5/20 0.83
AKR1B10 O60218 2/20 0.83
AKR1B1 P15121 2/20 0.83
CACNA1G O43497 2/20 0.83
CACNA1H O95180 2/20 0.83
MAOA P21397 1/20 0.83
PDE5A O76074 1/20 0.83
ACHE P22303 3/20 0.76
PTGS2 P35354 2/20 0.76
TP53 P04637 1/20 0.76
MDM2 Q00987 1/20 0.76
CYP3A4 P08684 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP2C19 P33261 1/20 0.70
PDPK1 O15530 1/20 0.68
PRKCA P17252 1/20 0.68
BACE1 P56817 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sophoraflavanone A SCHEMBL29624617 1.00 ABCG2 (1.00) ABCG2ESR1ESR2AKR1B10AKR1B1
Sophoraflavanone B SCHEMBL147316 0.91 ESR1 (1.00) ABCG2ESR1ESR2AKR1B10AKR1B1
Sophoraflavanone B SCHEMBL14304885 0.91 ESR1 (1.00) ABCG2ESR1ESR2AKR1B10AKR1B1
Sophoraflavanone B SCHEMBL29396586 0.91 ESR1 (1.00) ABCG2ESR1ESR2AKR1B10AKR1B1
Sophoraflavanone B SCHEMBL1171435 0.91 ESR1 (1.00) ABCG2ESR1ESR2AKR1B10AKR1B1
Sophoraflavanone B SCHEMBL1931652 0.90 ESR1 (0.98) ABCG2ESR1ESR2AKR1B10AKR1B1
SCHEMBL17626647 0.89 ABCG2 (0.79) ABCG2ESR1ESR2AKR1B10AKR1B1
SCHEMBL27013448 0.89 ABCG2 (0.79) ABCG2ESR1ESR2AKR1B10AKR1B1
SCHEMBL29808777 0.89 ABCG2 (0.79) ABCG2ESR1ESR2AKR1B10AKR1B1
SCHEMBL17626644 0.89 ABCG2 (0.79) ABCG2ESR1ESR2AKR1B10AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190046469-A1 COMPOSITIONS AND METHODS FOR TREATING MOOD DISORDERS OR SKIN DISEASE OR DAMAGE KUHRTS ERIC HAUSER (US) 2019-02-14 US claimed
US-20150209307-A1 COMPOSITIONS AND METHODS FOR TREATING MOOD DISORDERS OR SKIN DISEASE OR DAMAGE KUHRTS ERIC HAUSER (US) 2015-07-30 US claimed
WO-2014025989-A1 COMPOSITIONS AND METHODS FOR TREATING MOOD DISORDERS OR SKIN DISEASE OR DAMAGE KUHRTS ERIC HAUSER (US) 2014-02-13 WO claimed
US-20140045904-A1 NIACIN FORMULATIONS AND METHODS WITH REDUCED FLUSHING SIDE EFFECT KUHRTS ERIC HAUSER (US) 2014-02-13 US claimed
WO-2012051107-A2 NIACIN FORMULATIONS AND METHODS WITH REDUCED FLUSHING SIDE-EFFECT KUHRTS ERIC HAUSER (US) 2012-04-19 WO claimed
US-20120059052-A1 PRENYLFLAVONOID FORMULATIONS BIOACTIVES, INC. (US) 2012-03-08 US claimed
US-20110003888-A1 HOPS EXTRACTION METHODS AND MIXTURES BIOACTIVES, INC. (US) 2011-01-06 US claimed
US-20090209654-A1 Prenylflavonoid Formulations BIOACTIVES, INC. 2009-08-20 US claimed
WO-2008095189-A1 METHODS AND COMPOSITIONS FOR TREATING DYSLIPIDAEMIA BIOACTIVES, INC. (US) 2008-08-07 WO claimed
WO-2008089137-A1 HOPS EXTRACTION METHODS AND MIXTURES BIOACTIVES, INC. (US) 2008-07-24 WO claimed
EP-1909584-A2 PRENYLFLAVONOID FORMULATIONS Bioactives, Inc. (US) 2008-04-16 EP claimed
US-20070218155-A1 Methods and compositions for treating dyslipidaemia BIOACTIVES, INC. 2007-09-20 US claimed
WO-2007053915-A2 NARINGENIN DERIVATIVES WITH SELECTIVITY ON ERS UNIVERSITEIT GENT (BE) 2007-05-18 WO claimed
WO-2007016578-A2 PRENYLFLAVONOID FORMULATIONS BIOACTIVES, INC. (US) 2007-02-08 WO claimed
US-20050019438-A1 Hop extracts and use thereof in the production of a medicament having estrogenic properties BOURGES-SEVENIER CEDRIC (FR) 2005-01-27 US claimed
EP-1381379-A1 HOP EXTRACTS AND USE THEREOF IN THE PRODUCTION OF A MEDICAMENT HAVING ESTROGENIC PROPERTIES BERKEM (FR) 2004-01-21 EP claimed
WO-2002085393-A1 HOP EXTRACTS AND USE THEREOF IN THE PRODUCTION OF A MEDICAMENT HAVING ESTROGENIC PROPERTIES BERKEM (FR) 2002-10-31 WO claimed
US-20240091279-A1 COMBINATION THERAPY FOR INFLAMMATORY DISEASES NATIONAL INSTITUTES OF HEALTH 2024-03-21 US disclosed
WO-2003014287-A1 HOPS EXTRACTS, METHOD FOR THE PRODUCTION AND USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 2003-02-20 WO disclosed
WO-2002085393-A1 HOP EXTRACTS AND USE THEREOF IN THE PRODUCTION OF A MEDICAMENT HAVING ESTROGENIC PROPERTIES BERKEM (FR) 2002-10-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059052-A1 PRENYLFLAVONOID FORMULATIONS TP53, CYP46A1, HPGD ABCG2 110/4885ESR1 1771/4885ESR2 1616/4885
US-20150209307-A1 COMPOSITIONS AND METHODS FOR TREATING MOOD DISORDERS OR SKIN DISEASE OR DAMAGE CUTA, PSEN2, PNN ABCG2 4834/4885ESR1 421/4885ESR2 713/4885
US-20190046469-A1 COMPOSITIONS AND METHODS FOR TREATING MOOD DISORDERS OR SKIN DISEASE OR DAMAGE CUTA, PSEN2, PNN ABCG2 4834/4885ESR1 421/4885ESR2 713/4885
US-20110003888-A1 HOPS EXTRACTION METHODS AND MIXTURES HMGB2, HMGB3, HPGDS ABCG2 2079/4885ESR1 752/4885ESR2 599/4885
US-20140045904-A1 NIACIN FORMULATIONS AND METHODS WITH REDUCED FLUSHING SIDE EFFECT NAPRT, NISCH, NAMPT ABCG2 549/4885ESR1 2279/4885ESR2 3047/4885
US-20090209654-A1 Prenylflavonoid Formulations TP53, CYP46A1, HPGD ABCG2 110/4885ESR1 1771/4885ESR2 1616/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.