SCHEMBL14200327

SCHEMBL14200327

CCCCN(C(=O)CC(C)(C)C)c1ccc(C)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
PAX8 Q06710 2/20 0.46
JAK2 O60674 1/20 0.46
TP53 P04637 3/20 0.44
ALDH1A1 P00352 1/20 0.44
GPX4 P36969 1/20 0.44
MLYCD O95822 3/20 0.43
LTB4R2 Q9NPC1 1/20 0.39
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC1 Q13547 1/20 0.38
CNR2 P34972 1/20 0.37
OPRM1 P35372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200330 0.88 MLYCD (0.44) NPC1RAB9APAX8JAK2TP53
SCHEMBL14200342 0.88 NPC1 (0.47) NPC1RAB9APAX8JAK2TP53
SCHEMBL14200236 0.88 NPC1 (0.60) NPC1RAB9APAX8JAK2TP53
SCHEMBL14200760 0.86 NPC1 (0.46) NPC1RAB9APAX8JAK2TP53
SCHEMBL14200336 0.85 TRPM8 (0.45) NPC1RAB9APAX8JAK2ALDH1A1
SCHEMBL21549479 0.85 CNR2 (0.43) ALDH1A1MLYCDCNR2
SCHEMBL14200376 0.85 NPC1 (0.43) NPC1RAB9APAX8JAK2TP53
SCHEMBL14200332 0.84 ALDH1A1 (0.64) NPC1RAB9APAX8JAK2TP53
SCHEMBL8755638 0.83 NPC1 (0.67) NPC1RAB9APAX8JAK2TP53
SCHEMBL14174746 0.83 MLYCD (0.42) TP53ALDH1A1MLYCDMEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed