SCHEMBL14200439

SCHEMBL14200439

CCCCC(CCCC)N(C(=O)CC(C)(C)C)c1cccc(CC)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
EPHX1 P07099 1/20 0.37
CETP P11597 1/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SIGMAR1 Q99720 4/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200467 0.92 MAPK1 (0.37) MAPK1L3MBTL1EPHX1CETPTSHR
SCHEMBL14200451 0.91 PRKCA (0.36) EPHX1CETPALDH1A1CNR2PPARG
SCHEMBL14200452 0.87 SIGMAR1 (0.37) MAPK1L3MBTL1CETPTSHRTDP1
SCHEMBL14200442 0.87 MAPK1 (0.37) MAPK1L3MBTL1EPHX1TSHRTDP1
SCHEMBL14200503 0.86 ALDH1A1 (0.46) TDP1ALDH1A1SMN1; SMN2PPARGPPARA
SCHEMBL14229687 0.86 TP53 (0.40) MAPK1L3MBTL1EPHX1TSHRTDP1
SCHEMBL14200995 0.85 RIPK1 (0.39) L3MBTL1TSHRTDP1ALDH1A1SMN1; SMN2
SCHEMBL14200447 0.85 MAPK1 (0.36) MAPK1L3MBTL1EPHX1CETPTSHR
SCHEMBL14200444 0.85 ALDH1A1 (0.42) EPHX1ALDH1A1NPC1HPGD
SCHEMBL14200476 0.84 LTB4R2 (0.44) SMN1; SMN2NPC1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed