SCHEMBL14200516

SCHEMBL14200516

CCCCN(C(=O)CC(C)(C)C)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CETP P11597 5/20 0.45
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
PAX8 Q06710 2/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
GPX4 P36969 1/20 0.43
GRM2 Q14416 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
JAK2 O60674 1/20 0.39
LTB4R2 Q9NPC1 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
PPARG P37231 2/20 0.38
PPARA Q07869 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
MLYCD O95822 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229241 0.88 TP53 (0.49) CETPNPC1RAB9APAX8ALDH1A1
SCHEMBL14200337 0.87 MTNR1A (0.53) NPC1RAB9APAX8ALDH1A1TP53
SCHEMBL14200462 0.82 CETP (0.50) CETPGRM2PTGDR2PPARGPPARA
SCHEMBL14200328 0.82 LTB4R2 (0.49) CETPNPC1RAB9APAX8ALDH1A1
SCHEMBL14200332 0.80 ALDH1A1 (0.64) NPC1RAB9APAX8ALDH1A1TP53
SCHEMBL14200474 0.79 CETP (0.46) CETPGRM2PTGDR2PPARGPPARA
SCHEMBL14200338 0.79 ALDH1A1 (0.50) NPC1RAB9APAX8ALDH1A1TP53
SCHEMBL14200819 0.79 TP53 (0.47) NPC1RAB9APAX8ALDH1A1TP53
SCHEMBL14200463 0.79 CETP (0.48) CETPGRM2HDAC8
SCHEMBL14200475 0.79 CETP (0.46) CETPGRM2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed