SCHEMBL14200328

SCHEMBL14200328

CCCCN(C(=O)CC(C)(C)C)c1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 6/20 0.49
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
PAX8 Q06710 2/20 0.47
TP53 P04637 2/20 0.47
ALDH1A1 P00352 2/20 0.47
GPX4 P36969 1/20 0.47
JAK2 O60674 1/20 0.43
HDAC6 Q9UBN7 2/20 0.41
ACHE P22303 1/20 0.39
S1PR1 P21453 3/20 0.39
MLYCD O95822 1/20 0.39
RIPK1 Q13546 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
PTBP1 P26599 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CETP P11597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200332 0.85 ALDH1A1 (0.64) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14229341 0.85 LTB4R2 (0.58) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14200338 0.84 ALDH1A1 (0.50) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14200819 0.84 TP53 (0.47) NPC1RAB9APAX8TP53ALDH1A1
SCHEMBL14200330 0.83 MLYCD (0.44) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14200236 0.83 NPC1 (0.60) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14200572 0.83 TP53 (0.46) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14200574 0.83 NPC1 (0.48) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14200337 0.82 MTNR1A (0.53) LTB4R2NPC1RAB9APAX8TP53
SCHEMBL14200516 0.82 CETP (0.45) LTB4R2NPC1RAB9APAX8TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed