SCHEMBL14200780

SCHEMBL14200780

CCCCN(Cc1ccc(C)c(C)c1)C(=O)CC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 8/20 0.48
HDAC1 Q13547 7/20 0.48
HDAC3 O15379 2/20 0.48
HDAC2 Q92769 2/20 0.48
NCOR2 Q9Y618 1/20 0.48
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
LTB4R2 Q9NPC1 2/20 0.40
CNR2 P34972 3/20 0.39
SOAT1 P35610 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200898 0.92 HDAC1 (0.40) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14229430 0.85 HDAC6 (0.54) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14200916 0.83 GRIN2D (0.48) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14200848 0.83 TSHR (0.50) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14200903 0.83 RIPK1 (0.49) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14200828 0.81 HDAC3 (0.45) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14200343 0.81 CNR2 (0.54) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14200894 0.80 NPC1 (0.36) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL23992462 0.79 HDAC6 (0.51) HDAC6HDAC1HDAC3HDAC2NCOR2
SCHEMBL14200776 0.79 NPC1 (0.35) HDAC6HDAC1NPC1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed