SCHEMBL14200848

SCHEMBL14200848

CCCCN(Cc1ccc(Cl)c(Cl)c1)C(=O)CC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
HDAC1 Q13547 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
HDAC3 O15379 1/20 0.47
HDAC2 Q92769 1/20 0.47
NCOR2 Q9Y618 1/20 0.47
HSP90AA1 P07900 1/20 0.43
ALDH1A1 P00352 1/20 0.43
BLM P54132 1/20 0.43
CNR2 P34972 2/20 0.43
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200786 0.92 TSHR (0.41) TSHRHDAC1HDAC6HDAC3HDAC2
SCHEMBL14229228 0.85 TSHR (0.53) TSHRHDAC1HDAC6HDAC3HDAC2
SCHEMBL14200780 0.83 HDAC6 (0.48) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14200903 0.82 RIPK1 (0.49) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14200828 0.80 HDAC3 (0.45) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14200343 0.80 CNR2 (0.54) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14200916 0.80 GRIN2D (0.48) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14200849 0.79 PSEN1 (0.38) TSHRALDH1A1BLMSMN1; SMN2SIGMAR1
SCHEMBL23992462 0.78 HDAC6 (0.51) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229892 0.77 ALDH1A1 (0.47) TSHRHDAC1HDAC6HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed