SCHEMBL14200898

SCHEMBL14200898

CCCN(Cc1ccc(C)c(C)c1)C(=O)CC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
POLB P06746 1/20 0.39
APEX1 P27695 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
LMNA P02545 1/20 0.36
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
MLYCD O95822 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200780 0.92 HDAC6 (0.48) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229239 0.84 HDAC1 (0.44) HDAC1HDAC6POLBAPEX1TDP1
SCHEMBL14200852 0.82 RIPK1 (0.51) HDAC1HDAC6POLBAPEX1TDP1
SCHEMBL14200919 0.82 GRIN2D (0.46) HDAC1HDAC6POLBAPEX1TDP1
SCHEMBL14200786 0.82 TSHR (0.41) HDAC1HDAC6POLBAPEX1TDP1
SCHEMBL14200735 0.80 APP (0.47) LMNANPC1HPGDRAB9ATP53
SCHEMBL14200846 0.78 TAS1R3 (0.36) HDAC1HDAC6POLBLMNANPC1
SCHEMBL14200896 0.78 LMNA (0.36) HDAC1HDAC6POLBLMNANPC1
SCHEMBL14200765 0.77 TAS1R3 (0.36) HDAC1HDAC6POLBLMNANPC1
SCHEMBL14200827 0.77 TRPM8 (0.37) HDAC1HDAC6POLBLMNAS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed