SCHEMBL14201030

SCHEMBL14201030

CCCN(C(=O)CC(C)(C)C)c1ccc(F)c(Cl)c1F

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
ALDH1A1 P00352 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
FDFT1 P37268 5/20 0.32
MLYCD O95822 1/20 0.32
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
RIPK1 Q13546 2/20 0.31
P2RX7 Q99572 1/20 0.31
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14201040 0.92 ALDH1A1 (0.36) ALDH1A1FDFT1MLYCDTP53
SCHEMBL14229418 0.85 TP53 (0.42) LMNAALDH1A1NPSR1FDFT1MLYCD
SCHEMBL14228991 0.82 KDM4E (0.36) LMNAALDH1A1NPSR1MLYCDPOLB
SCHEMBL14201113 0.79 RIPK1 (0.32) FDFT1RIPK1
SCHEMBL14201021 0.78 RIPK1 (0.33) FDFT1RIPK1P2RX7
SCHEMBL14201018 0.78 PSEN1 (0.33) ALDH1A1FDFT1RIPK1
SCHEMBL14229898 0.77 TP53 (0.40) ALDH1A1MLYCDTP53
SCHEMBL14200873 0.77 RIPK1 (0.32) FDFT1RIPK1
SCHEMBL14201042 0.77 TSHR (0.31) FDFT1POLBRIPK1
SCHEMBL14200854 0.75 L3MBTL1 (0.34) ALDH1A1POLBAPEX1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed