SCHEMBL14201042

SCHEMBL14201042

CCCCC(CCCC)N(C(=O)CC(C)(C)C)c1ccc(F)c(Cl)c1F

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.31
RIPK1 Q13546 1/20 0.30
FDFT1 P37268 4/20 0.30
POLB P06746 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
MMP2 P08253 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14201113 0.93 RIPK1 (0.32) RIPK1FDFT1
SCHEMBL14201021 0.88 RIPK1 (0.33) RIPK1FDFT1
SCHEMBL14229417 0.87 TAS1R3 (0.31) TSHR
SCHEMBL14200872 0.86 MLYCD (0.33) MMP2
SCHEMBL14201018 0.85 PSEN1 (0.33) RIPK1FDFT1
SCHEMBL14200873 0.82 RIPK1 (0.32) RIPK1FDFT1
SCHEMBL14200471 0.80 ALDH1A1 (0.41) TSHRMMP2
SCHEMBL14200825 0.80 POLB (0.33) RIPK1POLB
SCHEMBL14201040 0.80 ALDH1A1 (0.36) TSHRFDFT1
SCHEMBL14229078 0.79 ALDH1A1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed